SCHEMBL8586368

SCHEMBL8586368

COc1ccc2c(c1)C(C#N)CCC2

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 1/20 0.47
KDM1A O60341 1/20 0.46
MAOA P21397 1/20 0.46
MAOB P27338 1/20 0.46
HTR2A P28223 1/20 0.46
HTR2C P28335 1/20 0.46
HTR2B P41595 1/20 0.46
MTNR1B P49286 2/20 0.45
GID4 Q8IVV7 1/20 0.45
MTNR1A P48039 2/20 0.44
SIGMAR1 Q99720 1/20 0.44
CYP19A1 P11511 3/20 0.44
CYP11B1 P15538 1/20 0.44
NQO2 P16083 1/20 0.44
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19469685 0.91 CYP19A1 (0.49) CHRNA7HTR2AHTR2CHTR2BMTNR1B
SCHEMBL9521714 0.88 CHRNA7 (0.47) CHRNA7HTR2CGID4SIGMAR1CYP19A1
SCHEMBL3161060 0.81 OPRM1 (0.44) HTR2AHTR2CHTR2BMTNR1BMTNR1A
SCHEMBL7439467 0.81 OPRM1 (0.44) HTR2AHTR2CHTR2BMTNR1BMTNR1A
SCHEMBL14199686 0.78 MTNR1A (0.53) MTNR1BMTNR1ASIGMAR1NQO2
SCHEMBL385632 0.78 CYP19A1 (0.49) CHRNA7HTR2CMTNR1BMTNR1ACYP19A1
SCHEMBL9814142 0.78 CHRNA7 (0.44) CHRNA7MAOAMEN1KMT2A
SCHEMBL13306289 0.78 HTR2C (0.62) CHRNA7KDM1AMAOAMAOBHTR2A
SCHEMBL29588202 0.78 HTR2C (0.62) CHRNA7KDM1AMAOAMAOBHTR2A
SCHEMBL2970487 0.78 HTR2C (0.62) CHRNA7KDM1AMAOAMAOBHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998052913-A2 LEUKOTRIENE B4 ANTAGONISTS, IN PARTICULAR 3-OXA-TETRAHYDRONAPHTHALENE-LTB4 ANTAGONISTS SCHERING AKTIENGESELLSCHAFT (DE) 1998-11-26 WO disclosed