SCHEMBL8587115

SCHEMBL8587115

CC(C)(C)OC(=O)NC(Cc1ccc(NC(N)=NC2CC2)s1)C(=O)OC(C)(C)C

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CTSS P25774 3/20 0.37
CTSK P43235 2/20 0.37
AAK1 Q2M2I8 1/20 0.36
CACNA1B Q00975 4/20 0.35
KMT2A Q03164 1/20 0.34
ITGB3 P05106 1/20 0.34
ITGB1 P05556 1/20 0.34
ITGAV P06756 1/20 0.34
ITGA2B P08514 1/20 0.34
ITGB5 P18084 1/20 0.34
MAPK1 P28482 1/20 0.34
SCN9A Q15858 1/20 0.33
TACR1 P25103 1/20 0.33
REN P00797 1/20 0.33
P2RY2 P41231 1/20 0.33
CTSL P07711 1/20 0.33
CTSB P07858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8529631 0.83 CTSS (0.43) CTSSCTSKTACR1P2RY2CTSL
SCHEMBL8529636 0.83 CTSS (0.43) CTSSCTSKTACR1P2RY2CTSL
SCHEMBL8526634 0.82 CTSS (0.36) CTSSCTSKAAK1ITGB3ITGB1
SCHEMBL8426516 0.79 ITGB3 (0.44) CTSSCTSKITGB3ITGB1ITGAV
SCHEMBL8530056 0.76 CTSS (0.45) CTSSCTSKAAK1TACR1P2RY2
SCHEMBL8422157 0.76 CTSS (0.45) CTSSCTSKTACR1P2RY2CTSL
SCHEMBL8530060 0.76 CTSS (0.45) CTSSCTSKAAK1TACR1P2RY2
SCHEMBL8422158 0.76 CTSS (0.45) CTSSCTSKTACR1P2RY2CTSL
SCHEMBL8422170 0.74 CTSS (0.45) CTSSCTSKITGB3ITGB1ITGAV
SCHEMBL8526061 0.74 ACE (0.45) CTSSCTSKITGB3ITGB1ITGAV

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0705257-B1 AMINOACID DERIVATIVES AS NO SYNTHASE INHIBITORS WELLCOME FOUND (GB) 1998-03-11 EP disclosed