SCHEMBL8587553

SCHEMBL8587553

COc1ccc(C(=O)Nc2cc(C3CCN(C)CC3)c[nH]2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.48
RAB9A P51151 1/20 0.48
CCNA2 P20248 1/20 0.47
CDK2 P24941 1/20 0.47
CCNA1 P78396 1/20 0.47
HDAC3 O15379 1/20 0.47
HDAC4 P56524 1/20 0.47
HDAC1 Q13547 1/20 0.47
HDAC7 Q8WUI4 1/20 0.47
HDAC2 Q92769 1/20 0.47
HDAC10 Q969S8 1/20 0.47
HDAC11 Q96DB2 1/20 0.47
HDAC8 Q9BY41 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
HDAC9 Q9UKV0 1/20 0.47
HDAC5 Q9UQL6 1/20 0.47
HTR1A P08908 2/20 0.46
HTR1F P30939 2/20 0.46
KDM1A O60341 2/20 0.46
MAOA P21397 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8636423 0.87 HTR1F (0.54) NPC1RAB9AHDAC3HDAC4HDAC1
SCHEMBL8639560 0.87 EPHX2 (0.45) NPC1RAB9AHDAC3HDAC4HDAC1
SCHEMBL8584266 0.86 HDAC3 (0.48) CCNA2CDK2CCNA1HDAC3HDAC4
SCHEMBL8586359 0.86 HTR1F (0.53) NPC1RAB9AHDAC3HDAC4HDAC1
SCHEMBL8586794 0.83 HTR1A (0.58) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL8584947 0.81 HTR1A (0.58) HTR1AHTR1FHTR1BHCN1
SCHEMBL8585175 0.81 HTR1A (0.46) NPC1RAB9AHTR1AHTR1FKDM1A
SCHEMBL8584756 0.78 HTR1D (0.51) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL8586100 0.77 HTR1D (0.41) HTR1AHTR1FPOLBALDH1A1HTR1D
SCHEMBL8587381 0.76 HTR1A (0.56) HDAC3HDAC4HDAC1HDAC7HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998020875-A1 5-HT1F AGONISTS ELI LILLY AND COMPANY (US) 1998-05-22 WO disclosed