SCHEMBL8587699

SCHEMBL8587699

CN(C)CCOc1cc(NC(=O)Nc2ccc(-c3ccncc3)c3ccccc23)ccc1I

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 2/20 0.43
KIT P10721 1/20 0.43
FLT3 P36888 1/20 0.43
ROCK2 O75116 3/20 0.42
ROCK1 Q13464 1/20 0.42
MCHR1 Q99705 1/20 0.42
HRH3 Q9Y5N1 3/20 0.41
GRM4 Q14833 1/20 0.40
KMT2A Q03164 1/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
NTRK1 P04629 1/20 0.39
AAK1 Q2M2I8 1/20 0.39
TNF P01375 1/20 0.39
HCK P08631 1/20 0.39
MAPK12 P53778 1/20 0.39
MAPK14 Q16539 1/20 0.39
HTR2C P28335 2/20 0.38
HTR2B P41595 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8588618 0.96 HRH3 (0.41) KDRKITFLT3ROCK2ROCK1
SCHEMBL8590672 0.95 KDR (0.45) KDRKITFLT3ROCK2ROCK1
SCHEMBL8589814 0.88 HRH3 (0.42) KDRKITFLT3ROCK2ROCK1
SCHEMBL8589856 0.86 HTR1D (0.47) KDRKITFLT3MCHR1HRH3
SCHEMBL8588968 0.85 MCHR1 (0.41) KDRKITFLT3ROCK2ROCK1
SCHEMBL8587765 0.83 HTR1D (0.44) MCHR1KMT2AKDM4EALDH1A1HTR2C
SCHEMBL8587717 0.82 RAB9A (0.53) HRH3KMT2AKDM4EALDH1A1SMN1; SMN2
SCHEMBL8591092 0.81 KDR (0.39) KDRKITFLT3ROCK2ROCK1
SCHEMBL8590131 0.79 MCHR1 (0.53) KDRKITFLT3MCHR1HRH3
SCHEMBL8617369 0.77 HTR1D (0.59) ROCK2ROCK1HTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998050346-A2 ACETAMIDE AND UREA DERIVATIVES, PROCESS FOR THEIR PREPARATION AND THEIR USE IN THE TREATMENT OF CNS DISORDERS SMITHKLINE BEECHAM PLC (GB) 1998-11-12 WO disclosed