SCHEMBL8587765

SCHEMBL8587765

CN(C)CCCc1cc(NC(=O)Nc2ccc(-c3ccncc3)c3ccccc23)ccc1I

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 4/20 0.44
HTR1B P28222 4/20 0.44
HTR1A P08908 2/20 0.44
ALDH1A1 P00352 2/20 0.44
MAPT P10636 2/20 0.44
TDP1 Q9NUW8 2/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
ALOX15 P16050 1/20 0.44
CYP2C19 P33261 1/20 0.44
IMPDH2 P12268 4/20 0.40
HTR2C P28335 2/20 0.38
HTR2B P41595 2/20 0.38
GAA P10253 2/20 0.38
DDX3X O00571 1/20 0.38
NAMPT P43490 1/20 0.37
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
KDM4E B2RXH2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8588618 0.86 HRH3 (0.41) HTR1DHTR1BCYP3A4CYP2D6IMPDH2
SCHEMBL8589654 0.85 HTR1D (0.44) HTR1DHTR1BHTR1AALDH1A1MAPT
SCHEMBL8587699 0.83 KDR (0.43) ALDH1A1IMPDH2HTR2CHTR2BKMT2A
SCHEMBL8590672 0.78 KDR (0.45) ALDH1A1IMPDH2KMT2AKDM4EMCHR1
SCHEMBL8613884 0.77 HTR1A (0.59) HTR1DHTR1BHTR1AALDH1A1MAPT
SCHEMBL8615090 0.76 HTR6 (0.49) HTR1DHTR1BHTR1AMAPTHTR2C
SCHEMBL8587499 0.74 MEN1 (0.54) MAPTCYP1A2MEN1KMT2ATRPV1
SCHEMBL8657486 0.72 KDM4C (0.38) HTR1DHTR1BHTR1AALDH1A1HTR2C
SCHEMBL8615837 0.71 POLB (0.39) HTR1DHTR1BHTR1AALDH1A1MAPT
SCHEMBL8589814 0.70 HRH3 (0.42) HTR1DHTR1BALDH1A1MAPTTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998050346-A2 ACETAMIDE AND UREA DERIVATIVES, PROCESS FOR THEIR PREPARATION AND THEIR USE IN THE TREATMENT OF CNS DISORDERS SMITHKLINE BEECHAM PLC (GB) 1998-11-12 WO claimed
WO-1998050346-A2 ACETAMIDE AND UREA DERIVATIVES, PROCESS FOR THEIR PREPARATION AND THEIR USE IN THE TREATMENT OF CNS DISORDERS SMITHKLINE BEECHAM PLC (GB) 1998-11-12 WO disclosed