SCHEMBL858838

SCHEMBL858838

CSCC(NC(=O)CCC(N)C(=O)O)C(=O)NCC(C)=O

nearest known ligand 0.59

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.59
GSTK1 Q9Y2Q3 1/20 0.59
GLO1 Q04760 2/20 0.55
NOD1 Q9Y239 9/20 0.46
FNTA P49354 2/20 0.42
FNTB P49356 2/20 0.42
PGGT1B P53609 1/20 0.42
FOLH1 Q04609 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14066343 1.00 PTGS1 (0.59) PTGS1GSTK1GLO1NOD1FNTA
S-Methylglutathione SCHEMBL13157330 0.91 PTGS1 (0.71) PTGS1GSTK1GLO1NOD1FNTA
S-Methylglutathione SCHEMBL1767370 0.91 PTGS1 (0.71) PTGS1GSTK1GLO1NOD1FNTA
S-Methylglutathione SCHEMBL13948109 0.91 PTGS1 (0.71) PTGS1GSTK1GLO1NOD1FNTA
S-Methylglutathione SCHEMBL1767369 0.91 PTGS1 (0.71) PTGS1GSTK1GLO1NOD1FNTA
SCHEMBL13853902 0.86 NOD1 (0.54) PTGS1GSTK1GLO1NOD1FNTA
SCHEMBL14538464 0.86 PTGS1 (0.55) PTGS1GSTK1GLO1NOD1FNTA
SCHEMBL677435 0.85 PTGS1 (0.80) PTGS1GSTK1GLO1NOD1FNTA
SCHEMBL13160954 0.85 PTGS1 (0.80) PTGS1GSTK1GLO1NOD1FNTA
SCHEMBL18813885 0.85 PTGS1 (0.41) PTGS1GSTK1GLO1NOD1FNTA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120238601-A1 TREATMENT OF CANCER BIPAR SCIENCES, INC. (US) 2012-09-20 US disclosed
US-8143447-B2 Benzamide precursor with sulfur substituent; poly-ADP-ribose polymerase inhibitors, antitumor agents; leukemia, breast, ovarian, lung, bladder, prostate, pancreatic, and cervical cancers BIPAR SCIENCES, INC. (US) 2012-03-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120238601-A1 TREATMENT OF CANCER PARP1, PARP2, PARP3 PTGS1 1042/4885GSTK1 917/4885GLO1 2118/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.