SCHEMBL8588698

SCHEMBL8588698

COc1ccc2nc3[nH]nc(-c4ccccc4)c3c(C)c2c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3A P49840 2/20 0.52
GSK3B P49841 2/20 0.52
AURKA O14965 2/20 0.47
CDK1 P06493 1/20 0.47
CDK4 P11802 1/20 0.47
CDK2 P24941 1/20 0.47
AKT1 P31749 1/20 0.47
KDM4E B2RXH2 6/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
MAPT P10636 4/20 0.46
TP53 P04637 2/20 0.46
PLA2G2A P14555 1/20 0.44
ALDH1A1 P00352 3/20 0.44
HSD17B10 Q99714 3/20 0.44
HPGD P15428 2/20 0.44
TSHR P16473 2/20 0.44
NPC1 O15118 1/20 0.44
NFKB1 P19838 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18079552 0.83 AURKA (0.52) AURKACDK1CDK4CDK2AKT1
SCHEMBL8591067 0.81 ELANE (0.39) GSK3AGSK3BKDM4EMAPTPLA2G2A
SCHEMBL9006232 0.73 AURKA (0.50) AURKACDK1CDK4CDK2AKT1
SCHEMBL4713601 0.72 BCHE (0.47) GSK3AGSK3BAURKACDK1CDK4
SCHEMBL24108922 0.72 KDM4E (0.55) KDM4ESMN1; SMN2MEN1KMT2AMAPT
SCHEMBL11705064 0.72 KDM4E (0.66) AURKAKDM4ESMN1; SMN2MEN1KMT2A
SCHEMBL11706523 0.71 MAPT (0.64) KDM4ESMN1; SMN2MEN1KMT2AMAPT
SCHEMBL1513055 0.71 CDK4 (0.60) GSK3AGSK3BCDK4CDK2KDM4E
SCHEMBL9006085 0.71 POLB (0.49) GSK3BAURKACDK1CDK4CDK2
SCHEMBL6591973 0.70 GSK3A (0.65) GSK3AGSK3BKDM4ESMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998049219-A1 PYRAZOL-BASED ELECTROLUMINESCENT POLYMERS AND THEIR USE IN ELECTROLUMINESCENT DEVICES THE UNIVERSITY COURT OF NAPIER UNIVERSITY (GB) 1998-11-05 WO disclosed