SCHEMBL8593268

SCHEMBL8593268

CCOC(=O)C(CCC(C#N)CCOC1CCCCO1)Cc1ccc(Cl)c(Cl)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 5/20 0.38
OPRK1 P41145 7/20 0.37
OPRM1 P35372 3/20 0.37
P2RX3 P56373 1/20 0.37
ALDH1A1 P00352 3/20 0.37
SMN1; SMN2 Q16637 3/20 0.37
KDM4E B2RXH2 1/20 0.37
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
SIGMAR1 Q99720 5/20 0.35
TSHR P16473 4/20 0.35
CYP2D6 P10635 3/20 0.35
TP53 P04637 2/20 0.35
CYP3A4 P08684 2/20 0.35
CYP1A2 P05177 2/20 0.35
CYP2C19 P33261 1/20 0.35
MTOR P42345 1/20 0.35
RAB9A P51151 1/20 0.35
OPRD1 P41143 1/20 0.35
MAPK8 P45983 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8590301 0.95 SLC6A3 (0.37) SLC6A3OPRK1OPRM1P2RX3ALDH1A1
SCHEMBL8290867 0.90 MEN1 (0.39) SLC6A3P2RX3ALDH1A1KDM4EMEN1
SCHEMBL8300283 0.80 MEN1 (0.40) SLC6A3P2RX3MEN1KMT2ASIGMAR1
SCHEMBL8592687 0.80 SLC6A3 (0.45) SLC6A3OPRK1OPRM1P2RX3MEN1
SCHEMBL8352398 0.80 SLC6A3 (0.45) SLC6A3OPRK1OPRM1SMN1; SMN2MEN1
SCHEMBL7496624 0.80 SLC6A3 (0.50) SLC6A3OPRK1OPRM1ALDH1A1SMN1; SMN2
SCHEMBL8556420 0.77 MEN1 (0.41) SLC6A3ALDH1A1KDM4EMEN1KMT2A
SCHEMBL4630703 0.72 SLC6A3 (0.45) SLC6A3MEN1KMT2ARAB9ASLC6A2
SCHEMBL8592295 0.72 MEN1 (0.38) SLC6A3OPRK1OPRM1P2RX3ALDH1A1
SCHEMBL6722595 0.72 MEN1 (0.54) MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5770735-A Polycyclic amine compounds and their enantiomers, their method of preparation and pharmaceutical compositions in which they are present ELF SANOFI (FR) 1998-06-23 US disclosed
US-5625060-A Polycyclic amine compounds and their enantiomers, their method of preparation and pharmaceutical compositions on which they are present Sanofi, Elf (FR) 1997-04-29 US disclosed
US-5340822-A Substance P, neurokinin antagonists ELF SANOFI (FR) 1994-08-23 US disclosed