SCHEMBL8595641

SCHEMBL8595641

CCCCc1nc(CCc2ccccc2)[nH]c(=O)c1Cc1ccc(Br)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.45
MAPT P10636 2/20 0.43
ALDH1A1 P00352 1/20 0.43
HPGD P15428 1/20 0.43
POLB P06746 2/20 0.42
KMT2A Q03164 2/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
RNASEH1 O60930 1/20 0.41
DAO P14920 2/20 0.40
TUBB4A P04350 1/20 0.40
TUBB P07437 1/20 0.40
TUBA3C P0DPH7 1/20 0.40
TUBA1B P68363 1/20 0.40
TUBA4A P68366 1/20 0.40
TUBB4B P68371 1/20 0.40
TUBB3 Q13509 1/20 0.40
TUBB2A Q13885 1/20 0.40
TUBB8 Q3ZCM7 1/20 0.40
TUBA3E Q6PEY2 1/20 0.40
TUBA1A Q71U36 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27771388 0.90 PARP1 (0.46) PARP1MAPTALDH1A1HPGDPOLB
SCHEMBL1886429 0.82 ACHE (0.43) PARP1
SCHEMBL8670123 0.80 HIF1A (0.49) MAPTALDH1A1HPGDKMT2AMEN1
SCHEMBL9257694 0.80
SCHEMBL1895574 0.79 PPARG (0.52)
SCHEMBL27771406 0.79 ALDH1A1 (0.44) PARP1MAPTALDH1A1HPGDPOLB
SCHEMBL27771413 0.78 BRS3 (0.39) PARP1MAPTALDH1A1HPGDTUBB4A
SCHEMBL28236562 0.78 ALDH1A1 (0.50) PARP1MAPTALDH1A1HPGDPOLB
SCHEMBL9129778 0.76
SCHEMBL9196627 0.75 AGTR1 (0.55)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0593332-B1 Phenylborinic acid derivatives, their preparation and their use as intermediates in syntheses SYNTHELABO (FR) 1998-01-14 EP disclosed
EP-0655452-A1 Triarylborane derivatives, their preparation and their use as intermediates SYNTHELABO (FR) 1995-05-31 EP disclosed
US-5405960-A Triarylborane derivatives, their preparation and their use as synthesis intermediates SYNTHELABO (FR) 1995-04-11 US disclosed
US-5382672-A Preparation of derivatives of benzeneborinic acid SYNTHELABO (FR) 1995-01-17 US disclosed
US-5374735-A Triarylborane derivatives, their preparation and their use as synthesis intermediates SYNTHELABO (FR) 1994-12-20 US disclosed
US-5312920-A Process for preparing 4-pyrimidinones SYNTHELABO (FR) 1994-05-17 US disclosed
EP-0593332-A1 Phenylboronic acid derivatives, their preparation and their use as intermediates in syntheses SYNTHELABO (FR) 1994-04-20 EP disclosed
US-5278312-A Derivatives of benzeneborinic acid, preparation thereof and use thereof as synthetic intermediates SYNTHELABO (FR) 1994-01-11 US disclosed
EP-0561664-A1 Process for the preparation of 4-pyrimidines SYNTHELABO (FR) 1993-09-22 EP disclosed