SCHEMBL8596190

SCHEMBL8596190

CC=CCC1Cc2ccc(O)cc2C1=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 2/20 0.43
METAP1 P53582 4/20 0.42
MEN1 O00255 2/20 0.40
GLA P06280 2/20 0.40
KMT2A Q03164 2/20 0.40
GAA P10253 1/20 0.40
KDM4E B2RXH2 1/20 0.40
NPC1 O15118 1/20 0.40
NR1I2 O75469 1/20 0.40
GMNN O75496 1/20 0.40
USP2 O75604 1/20 0.40
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
TP53 P04637 1/20 0.40
CYP1A2 P05177 1/20 0.40
HSP90AA1 P07900 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
MAPT P10636 1/20 0.40
CYP2C9 P11712 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8874593 1.00 CYP19A1 (0.43) CYP19A1METAP1MEN1GLAKMT2A
SCHEMBL8596188 1.00 CYP19A1 (0.43) CYP19A1METAP1MEN1GLAKMT2A
SCHEMBL8874447 0.86 METAP1 (0.47) METAP1PBRM1ACHE
SCHEMBL8600861 0.86 METAP1 (0.47) METAP1PBRM1ACHE
SCHEMBL8600862 0.86 METAP1 (0.47) METAP1PBRM1ACHE
SCHEMBL8873299 0.84 METAP1 (0.59) METAP1ACHE
SCHEMBL8595392 0.84 METAP1 (0.59) METAP1ACHE
SCHEMBL8595390 0.84 METAP1 (0.59) METAP1ACHE
SCHEMBL8873173 0.83 ACHE (0.55) METAP1ACHE
SCHEMBL8595937 0.83 METAP1 (0.47) METAP1MAOBACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0657426-B1 Tricyclic pyrrole derivatives HOFFMANN LA ROCHE (CH) 1998-07-22 EP disclosed
US-5646173-A ANTISEROTONINE AGENTS; CENTRAL NERVOUS SYSTEM DISORDERS; ANTIDEPRESSANTS HOFFMANN-LA ROCHE INC. (US) 1997-07-08 US disclosed
EP-0657426-A2 Tricyclic pyrrole derivatives F. HOFFMANN-LA ROCHE AG (CH) 1995-06-14 EP disclosed