SCHEMBL8596238

SCHEMBL8596238

COc1ccc2ccc3ccn(C[C@H](C)N)c3c2c1

nearest known ligand 0.66

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 19/20 0.66
HTR2A P28223 17/20 0.63
HTR2B P41595 5/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8596900 1.00 HTR2C (0.66) HTR2CHTR2AHTR2B
Fumaric Acid SCHEMBL8874855 0.89 HTR2C (0.54) HTR2CHTR2AHTR2B
Fumaric Acid SCHEMBL8873561 0.89 HTR2C (0.54) HTR2CHTR2AHTR2B
Fumaric Acid SCHEMBL8873554 0.89 HTR2C (0.54) HTR2CHTR2AHTR2B
Fumaric Acid SCHEMBL8874862 0.89 HTR2C (0.54) HTR2CHTR2AHTR2B
SCHEMBL7093740 0.81 HTR2C (0.81) HTR2CHTR2AHTR2B
SCHEMBL7997598 0.81 HTR2C (0.81) HTR2CHTR2AHTR2B
SCHEMBL8874209 0.80 HTR2C (0.46) HTR2CHTR2A
SCHEMBL6365952 0.76 HTR2C (0.70) HTR2CHTR2AHTR2B
SCHEMBL7767788 0.76 HTR2C (0.70) HTR2CHTR2AHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0657426-B1 Tricyclic pyrrole derivatives HOFFMANN LA ROCHE (CH) 1998-07-22 EP claimed
US-5646173-A ANTISEROTONINE AGENTS; CENTRAL NERVOUS SYSTEM DISORDERS; ANTIDEPRESSANTS HOFFMANN-LA ROCHE INC. (US) 1997-07-08 US claimed
EP-0657426-A2 Tricyclic pyrrole derivatives F. HOFFMANN-LA ROCHE AG (CH) 1995-06-14 EP claimed
EP-0657426-B1 Tricyclic pyrrole derivatives HOFFMANN LA ROCHE (CH) 1998-07-22 EP disclosed
US-5646173-A ANTISEROTONINE AGENTS; CENTRAL NERVOUS SYSTEM DISORDERS; ANTIDEPRESSANTS HOFFMANN-LA ROCHE INC. (US) 1997-07-08 US disclosed
EP-0657426-A2 Tricyclic pyrrole derivatives F. HOFFMANN-LA ROCHE AG (CH) 1995-06-14 EP disclosed