SCHEMBL8597809

SCHEMBL8597809

COC(=N)c1c(F)cccc1F

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.44
CES1 P23141 2/20 0.44
RAB9A P51151 2/20 0.41
POLB P06746 2/20 0.40
KMT2A Q03164 4/20 0.38
MEN1 O00255 1/20 0.37
NPC1 O15118 1/20 0.36
CYP1A2 P05177 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
KRAS P01116 1/20 0.36
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA7 P43166 1/20 0.35
CA9 Q16790 1/20 0.35
CA14 Q9ULX7 1/20 0.35
JAK2 O60674 1/20 0.35
JAK1 P23458 1/20 0.35
TYK2 P29597 1/20 0.35
HTT P42858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27451039 0.82 CES2 (0.34) CES2CES1RAB9APOLBKMT2A
SCHEMBL8299666 0.77 NLRP3 (0.41) CES2CES1RAB9APOLBKMT2A
SCHEMBL8784070 0.76 GAA (0.48) CES2CES1RAB9AKMT2AMEN1
SCHEMBL1070351 0.73 CA12 (0.61) CES2CES1RAB9APOLBKMT2A
SCHEMBL4478269 0.72 NPC1 (0.50) CES2CES1RAB9AKMT2AMEN1
Iodide SCHEMBL6190800 0.71 CES2 (0.48) CES2CES1POLBKMT2AMEN1
SCHEMBL17063994 0.71 KMT2A (0.48) RAB9APOLBKMT2ANPC1TDP1
SCHEMBL642257 0.70 CES2 (0.46) CES2CES1RAB9AKMT2AMEN1
SCHEMBL10441887 0.70 CES2 (0.64) CES2CES1RAB9APOLBKMT2A
SCHEMBL14333527 0.69 CES2 (0.50) CES2CES1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0821677-A1 OXAZOLINE AND THIAZOLINE ARTHROPODICIDES E.I. DU PONT DE NEMOURS AND COMPANY (US) 1998-02-04 EP disclosed
EP-0741714-A1 ARTHROPODICIDAL 2-OXA AND THIA-ZOLINES E.I. DU PONT DE NEMOURS AND COMPANY (US) 1996-11-13 EP disclosed
WO-1996033180-A1 OXAZOLINE AND THIAZOLINE ARTHROPODICIDES E.I. DU PONT DE NEMOURS AND COMPANY (US) 1996-10-24 WO disclosed
WO-1995019972-A1 ARTHROPODICIDAL 2-OXA AND THIA-ZOLINES E.I. DU PONT DE NEMOURS AND COMPANY (US) 1995-07-27 WO disclosed