SCHEMBL8598142

SCHEMBL8598142

C=CCOc1ccc(-c2cc(C#CCCCC(C)F)ccc2-c2cccnc2)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 3/20 0.38
CYP2D6 P10635 2/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
GBA1 P04062 1/20 0.37
CYP11B1 P15538 4/20 0.33
CYP11B2 P19099 4/20 0.33
MGAM O43451 3/20 0.33
GAA P10253 3/20 0.33
SI P14410 3/20 0.33
MGAM2 Q2M2H8 3/20 0.33
MAPT P10636 2/20 0.33
GRM5 P41594 1/20 0.33
NPC1 O15118 1/20 0.33
HTT P42858 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
PTAFR P25105 3/20 0.33
CYP17A1 P05093 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8601722 0.90 MGAM (0.33) CYP2D6MGAMGAASIMGAM2
SCHEMBL8601450 0.89 CYP11B1 (0.41) CYP19A1CYP3A4GBA1CYP11B1CYP11B2
SCHEMBL8598099 0.88 CYP2D6 (0.38) CYP19A1CYP2D6CYP2C9CYP2C19MGAM
SCHEMBL8602104 0.88 PTAFR (0.37) CYP19A1CYP2D6CYP3A4CYP2C9CYP2C19
SCHEMBL8601719 0.85 DCTPP1 (0.33) MGAMGAASIMGAM2
SCHEMBL8600391 0.82 PTAFR (0.40) CYP19A1CYP2D6CYP3A4CYP2C9CYP2C19
SCHEMBL8600956 0.82 PTAFR (0.40) CYP19A1CYP2D6CYP3A4CYP2C9CYP2C19
SCHEMBL8599406 0.81 CYP19A1 (0.36) CYP19A1CYP2D6CYP3A4CYP2C9CYP2C19
SCHEMBL8604072 0.80 CYP2D6 (0.40) CYP2D6MGAMGAASIMGAM2
SCHEMBL7561123 0.80 CYP2D6 (0.40) CYP2D6MGAMGAASIMGAM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5779934-A FLUORINATING AN ALCOHOL DERIVATIVE SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1998-07-14 US disclosed