SCHEMBL8601450

SCHEMBL8601450

C=CCOc1cc(C#CCCCC(C)F)ccc1-c1cccnc1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 10/20 0.41
CYP11B2 P19099 10/20 0.41
CYP19A1 P11511 4/20 0.41
AAK1 Q2M2I8 1/20 0.35
MKNK1 Q9BUB5 1/20 0.35
MKNK2 Q9HBH9 1/20 0.35
GRM5 P41594 1/20 0.35
POLB P06746 1/20 0.34
GBA1 P04062 1/20 0.34
CHRNB2 P17787 1/20 0.34
CHRNA4 P43681 1/20 0.34
CYP17A1 P05093 1/20 0.33
CYP3A4 P08684 1/20 0.33
PTAFR P25105 1/20 0.33
ERN1 O75460 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8598478 0.89 AAK1 (0.32) AAK1CHRNB2CHRNA4
SCHEMBL8598142 0.89 CYP19A1 (0.38) CYP11B1CYP11B2CYP19A1GRM5POLB
SCHEMBL8600956 0.85 PTAFR (0.40) CYP11B1CYP11B2CYP19A1AAK1GRM5
SCHEMBL8602211 0.82 ERN1 (0.33) ERN1
SCHEMBL8602621 0.82 SQOR (0.31)
SCHEMBL8601156 0.82 CYP2D6 (0.32) CYP19A1
SCHEMBL8602104 0.81 PTAFR (0.37) CYP11B1CYP11B2CYP19A1MKNK1MKNK2
SCHEMBL8600165 0.81 FGFR4 (0.36)
SCHEMBL8604338 0.81 CYP11B1 (0.42) CYP11B1CYP11B2CYP19A1AAK1POLB
SCHEMBL8597829 0.79 CYP11B1 (0.38) CYP11B1CYP11B2CYP19A1AAK1MKNK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5779934-A FLUORINATING AN ALCOHOL DERIVATIVE SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1998-07-14 US disclosed