SCHEMBL8602104

SCHEMBL8602104

C=CCc1ccc(-c2cc(C#CCCCC(C)F)ccc2-c2cccnc2)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTAFR P25105 5/20 0.37
GRM5 P41594 1/20 0.34
MKNK1 Q9BUB5 1/20 0.33
MKNK2 Q9HBH9 1/20 0.33
CHRNB2 P17787 3/20 0.33
CHRNA4 P43681 3/20 0.33
CYP11B1 P15538 2/20 0.32
CYP11B2 P19099 2/20 0.32
CYP19A1 P11511 2/20 0.32
GBA1 P04062 1/20 0.32
AKR1C3 P42330 1/20 0.31
AKR1C2 P52895 1/20 0.31
ACE2 Q9BYF1 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
PPARG P37231 1/20 0.31
PPARA Q07869 1/20 0.31
PTGS2 P35354 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8599898 0.90
SCHEMBL8598142 0.88 CYP19A1 (0.38) PTAFRGRM5CHRNB2CHRNA4CYP11B1
SCHEMBL8600956 0.87 PTAFR (0.40) PTAFRGRM5CHRNB2CHRNA4CYP11B1
SCHEMBL8598924 0.85
SCHEMBL8603103 0.82 PTAFR (0.43) PTAFRMKNK1MKNK2AKR1C3AKR1C2
SCHEMBL8601450 0.81 CYP11B1 (0.41) PTAFRGRM5MKNK1MKNK2CHRNB2
SCHEMBL8599353 0.79 PTAFR (0.37) PTAFRMKNK1MKNK2CHRNB2CHRNA4
SCHEMBL8604574 0.79 ALDH1A1 (0.33) CYP3A4PTGS2
SCHEMBL7559816 0.79 ALDH1A1 (0.33) CYP3A4PTGS2
SCHEMBL8601722 0.77 MGAM (0.33) CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5779934-A FLUORINATING AN ALCOHOL DERIVATIVE SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1998-07-14 US disclosed