SCHEMBL8599298

SCHEMBL8599298

COc1ccc2cc(C3CCC(=O)CC3)sc2c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 1/20 0.47
PDE3B Q13370 2/20 0.41
PDE3A Q14432 2/20 0.41
CHRNA7 P36544 3/20 0.41
HTR1A P08908 3/20 0.41
MPI P34949 1/20 0.39
ALK Q9UM73 1/20 0.38
SLC6A4 P31645 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C19 P33261 1/20 0.37
MAOA P21397 1/20 0.37
MAOB P27338 1/20 0.37
PDE4A P27815 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE4C Q08493 1/20 0.36
PDE4D Q08499 1/20 0.36
ALDH1A1 P00352 2/20 0.36
GSTP1 P09211 1/20 0.36
PDK1 Q15118 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4450281 0.85 CA2 (0.48) CA2CHRNA7HTR1AMPISLC6A4
SCHEMBL8601229 0.84 CA2 (0.47) CA2CHRNA7HTR1AMPISLC6A4
SCHEMBL4438841 0.84 CA2 (0.47) CA2CHRNA7HTR1AMPISLC6A4
SCHEMBL4442739 0.84 CA2 (0.47) CA2CHRNA7HTR1AMPISLC6A4
SCHEMBL4442733 0.84 CA2 (0.47) CA2CHRNA7HTR1AMPISLC6A4
SCHEMBL4442755 0.84 CA2 (0.47) CA2CHRNA7HTR1AMPISLC6A4
SCHEMBL4444144 0.82 CA2 (0.46) CA2PDE3BPDE3ACHRNA7HTR1A
SCHEMBL6311284 0.81 HTR2C (0.50) CA2PDE3BPDE3ACHRNA7HTR1A
Water SCHEMBL7870821 0.80 HTR2C (0.49) CA2PDE3BPDE3ACHRNA7HTR1A
SCHEMBL8601033 0.77 HTR1A (0.41) CA2CHRNA7HTR1AMPISLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0641791-B1 NOVEL BENZOTHIOPHENE DERIVATIVE TEIKOKU HORMONE MFG CO LTD (JP) 1998-01-28 EP disclosed
US-5472962-A Antiestrogenic agents TEIKOKU HORMONE MFG. CO., LTD. (JP) 1995-12-05 US disclosed
EP-0641791-A1 NOVEL BENZOTHIOPHENE DERIVATIVE TEIKOKU HORMONE MFG. CO., LTD. (JP) 1995-03-08 EP disclosed