SCHEMBL8599580

SCHEMBL8599580

Clc1ccnc2cc(Cc3ccccc3)ccc12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.47
KDM4E B2RXH2 2/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C19 P33261 1/20 0.41
HIF1A Q16665 1/20 0.41
IDH1 O75874 1/20 0.40
MEN1 O00255 2/20 0.39
MAPT P10636 2/20 0.39
KMT2A Q03164 2/20 0.39
TDP1 Q9NUW8 2/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
CCNC P24863 1/20 0.39
CDK8 P49336 1/20 0.39
CALM1 P0DP23 1/20 0.39
CHKA P35790 1/20 0.38
LTA4H P09960 1/20 0.38
PTGES O14684 1/20 0.38
CYP2C9 P11712 1/20 0.38
TSHR P16473 1/20 0.38
MAPK1 P28482 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3871113 0.81 IDH1 (0.51) PKMIDH1CALM1CYP2C9KDM4A
SCHEMBL4387604 0.78 NR4A2 (0.40) PKMKDM4EMEN1MAPTKMT2A
SCHEMBL28175236 0.78 NR4A2 (0.40) PKMKDM4EMEN1MAPTKMT2A
SCHEMBL4389974 0.78 RECQL (0.52) PKMKDM4EMEN1MAPTKMT2A
SCHEMBL5519979 0.78 LOXL2 (0.52) NR4A2SOS2ROCK1
SCHEMBL30471785 0.78 NR4A2 (0.40) PKMKDM4EMEN1MAPTKMT2A
SCHEMBL29878333 0.77 CYP3A4 (0.58) PKMCYP3A4CYP2C19HIF1ALMNA
SCHEMBL3898712 0.77 CYP3A4 (0.58) PKMCYP3A4CYP2C19HIF1ALMNA
SCHEMBL5531943 0.77 NR4A2 (0.39) PKMCYP2C19MEN1MAPTKMT2A
SCHEMBL27956165 0.76 CA2 (0.50) KDM4EHIF1AMEN1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5773449-A BACTERICIDES FOR HELICOBACTER ZENYAKU KOGYO KABUSHIKI KAISHA (JP) 1998-06-30 US disclosed
EP-0786454-A1 THIOQUINOLONE DERIVATIVE ZENYAKU KOGYO KABUSHIKIKAISHA (JP) 1997-07-30 EP disclosed