SCHEMBL8600276

SCHEMBL8600276

C=CCN(CC=C)C(=O)c1c([N+](=O)[O-])c(N)nc2ccccc12

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.40
HPGD P15428 2/20 0.40
MAPT P10636 5/20 0.38
CDK5 Q00535 1/20 0.37
CDK5R1 Q15078 1/20 0.37
POLB P06746 2/20 0.36
MGMT P16455 1/20 0.36
LMNA P02545 3/20 0.35
MAPK1 P28482 2/20 0.35
KMT2A Q03164 3/20 0.35
KDM4E B2RXH2 5/20 0.35
HTT P42858 2/20 0.35
GSK3A P49840 1/20 0.35
GSK3B P49841 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
ATM Q13315 1/20 0.33
MEN1 O00255 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8598395 0.84 ALDH1A1 (0.40) ALDH1A1HPGDMAPTPOLBLMNA
SCHEMBL8601173 0.82 ALDH1A1 (0.42) ALDH1A1HPGDMAPTCDK5CDK5R1
SCHEMBL8599626 0.80 HPGD (0.50) ALDH1A1HPGDMAPTCDK5CDK5R1
SCHEMBL8568375 0.79 PDE10A (0.46) ALDH1A1MAPTCDK5CDK5R1MGMT
SCHEMBL8596169 0.79 MAPT (0.41) ALDH1A1HPGDMAPTCDK5CDK5R1
SCHEMBL8559921 0.78 IKBKB (0.42) ALDH1A1MAPTCDK5CDK5R1POLB
SCHEMBL8597641 0.77 KDM4E (0.41) ALDH1A1HPGDMAPTPOLBLMNA
SCHEMBL8568405 0.76 HSD17B10 (0.52) ALDH1A1HPGDMAPTCDK5CDK5R1
SCHEMBL8596304 0.75 MAPT (0.38) ALDH1A1HPGDMAPTCDK5CDK5R1
SCHEMBL8564023 0.75 MAPT (0.44) ALDH1A1HPGDMAPTCDK5CDK5R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0735025-B1 Process for producing aminonitropyridines SUMITOMO CHEMICAL CO (JP) 1998-07-01 EP disclosed
US-5648496-A AMINATION SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1997-07-15 US disclosed
EP-0735025-A1 Process for producing aminonitropyridines SUMITOMO CHEMICAL COMPANY LIMITED (JP) 1996-10-02 EP disclosed