SCHEMBL8602385

SCHEMBL8602385

COc1ccc(S(=O)(=O)n2ncc3ccccc3c2=O)cc1OC

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 5/20 0.63
PDE4B Q07343 5/20 0.63
PDE4C Q08493 5/20 0.63
PDE4D Q08499 5/20 0.63
HCRTR1 O43613 1/20 0.47
CYP2D6 P10635 1/20 0.47
MAPT P10636 2/20 0.46
KDM4E B2RXH2 1/20 0.46
ALDH1A1 P00352 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
KEAP1 Q14145 1/20 0.45
NFE2L2 Q16236 1/20 0.45
CTSG P08311 1/20 0.45
CMA1 P23946 1/20 0.45
HTR6 P50406 1/20 0.44
GPBAR1 Q8TDU6 1/20 0.44
USP2 O75604 1/20 0.44
LMNA P02545 1/20 0.44
GLA P06280 1/20 0.44
TSHR P16473 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31051613 0.84 CA12 (0.46) PDE4APDE4BPDE4CPDE4DMAPT
SCHEMBL30375363 0.79 CA12 (0.50) KDM4EALDH1A1TDP1HTR6LMNA
SCHEMBL7359664 0.78 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DHCRTR1
SCHEMBL7360978 0.74 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DHCRTR1
SCHEMBL7392643 0.72 PDE4A (0.66) PDE4APDE4BPDE4CPDE4DHCRTR1
SCHEMBL11318137 0.71 KMT2A (0.52) MAPTKDM4EALDH1A1USP2MAPK1
SCHEMBL7358727 0.71 PDE4A (0.67) PDE4APDE4BPDE4CPDE4DMAPT
SCHEMBL13633829 0.70 GAA (0.63) MAPTALDH1A1USP2LMNATSHR
SCHEMBL7366201 0.69 PDE4A (0.62) PDE4APDE4BPDE4CPDE4DMAPT
SCHEMBL7362713 0.68 PDE4A (0.63) PDE4APDE4BPDE4CPDE4DMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5728712-A 3,4-disubstituted-phenylsulphonamides and their therapeutic use CHIROSCIENCE LIMITED (GB) 1998-03-17 US disclosed