SCHEMBL8604584

SCHEMBL8604584

CC(C)(C)OC(=O)NCCc1ccc(OCCC2Oc3ccccc3N(Cc3cccc(Cl)c3)C2=O)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.45
TSHR P16473 1/20 0.44
ALDH1A1 P00352 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
TP53 P04637 3/20 0.42
XIAP P98170 1/20 0.41
FNTA P49354 1/20 0.40
FNTB P49356 1/20 0.40
PGGT1B P53609 1/20 0.40
MAPT P10636 2/20 0.39
SLC5A1 P13866 1/20 0.38
PPARG P37231 2/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
MAPK1 P28482 1/20 0.38
CYP2C19 P33261 1/20 0.38
HDAC2 Q92769 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8603793 0.93 ALDH1A1 (0.45) TSHRALDH1A1SMN1; SMN2TP53XIAP
SCHEMBL8604456 0.92 TSHR (0.45) KDM4ETSHRALDH1A1SMN1; SMN2TP53
SCHEMBL8605054 0.90 TSHR (0.43) TSHRALDH1A1SMN1; SMN2TP53MAPT
SCHEMBL8554618 0.90 KDM4E (0.41) KDM4ETSHRALDH1A1SMN1; SMN2TP53
SCHEMBL8551614 0.90 TSHR (0.43) TSHRALDH1A1SMN1; SMN2TP53MAPT
SCHEMBL8552315 0.89 TSHR (0.43) TSHRALDH1A1SMN1; SMN2TP53XIAP
SCHEMBL8604513 0.88 TSHR (0.44) TSHRALDH1A1SMN1; SMN2TP53SLC5A1
SCHEMBL8554097 0.88 ALDH1A1 (0.45) TSHRALDH1A1SMN1; SMN2TP53PPARG
SCHEMBL8603405 0.86 TSHR (0.42) TSHRALDH1A1SMN1; SMN2TP53XIAP
SCHEMBL8554119 0.85 TSHR (0.43) TSHRALDH1A1SMN1; SMN2TP53XIAP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5854242-A Benzoxazine antimicrobial agents ORTHO PHARMACEUTICAL CORPORATION (US) 1998-12-29 US disclosed
US-5696117-A BACTERICIDE ORTHO PHARMACEUTICAL CORPORATION (US) 1997-12-09 US disclosed