SCHEMBL8604971

SCHEMBL8604971

COc1cc(OC)c2[nH]cc(C3=C(O)C(=O)C(c4c[nH]c5c(OC)cc(OC)cc45)=C(O)C3=O)c2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 2/20 0.46
MTNR1B P49286 2/20 0.46
NQO2 P16083 2/20 0.43
CYP3A4 P08684 2/20 0.43
ALDH1A1 P00352 2/20 0.43
CYP1A2 P05177 1/20 0.43
ME2 P23368 1/20 0.40
ME1 P48163 1/20 0.40
ME3 Q16798 1/20 0.40
KDR P35968 2/20 0.39
ELANE P08246 2/20 0.39
CDK4 P11802 1/20 0.38
CCND1 P24385 1/20 0.38
CYP19A1 P11511 1/20 0.35
USP2 O75604 1/20 0.35
MAPK1 P28482 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
ERN1 O75460 1/20 0.35
ACHE P22303 1/20 0.35
KDM4E B2RXH2 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8604209 0.78 EGFR (0.44) CYP3A4ALDH1A1CYP1A2ME2ME1
SCHEMBL8604085 0.72 CNR1 (0.39) NQO2ALDH1A1ME2ME1ME3
SCHEMBL30353206 0.70 KDM4E (0.64) MTNR1AMTNR1BNQO2ALDH1A1CYP1A2
SCHEMBL21712157 0.69 MTNR1A (0.52) MTNR1AMTNR1BNQO2CYP3A4ALDH1A1
SCHEMBL3210719 0.69 ALDH1A1 (0.56) MTNR1AMTNR1BNQO2CYP3A4ALDH1A1
SCHEMBL6095610 0.68 ALDH1A1 (0.47) MTNR1AMTNR1BNQO2CYP3A4ALDH1A1
SCHEMBL8578397 0.68 MTNR1A (0.63) MTNR1AMTNR1BNQO2ALDH1A1KDM4E
SCHEMBL7291800 0.67 NQO2 (0.50) MTNR1AMTNR1BNQO2CYP3A4ALDH1A1
SCHEMBL5822130 0.66 ALDH1A1 (0.73) CYP3A4ALDH1A1CYP1A2ELANEUSP2
SCHEMBL6096465 0.65 KDR (0.50) MTNR1AMTNR1BCYP3A4ALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5786488-A DEHYDROBROMINATION OF A DIBROMOBENZOQUINONES WITH AT LEAST ONE INDOLES IN A POLAR SOLVENT AND A METAL CARBONATE TO FORM AN ANTITUMOR AGENT SUGEN, INC. (US) 1998-07-28 US disclosed
US-5780496-A Method and compositions for inhibition of adaptor protein/tyrosine kinase interactions SUGEN, INC. (US) 1998-07-14 US disclosed