SCHEMBL8604085

SCHEMBL8604085

COc1ccc(OC)c2c(C3=C(O)C(=O)C(c4c[nH]c5c(OC)ccc(OC)c45)=C(O)C3=O)c[nH]c12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 1/20 0.39
CNR2 P34972 1/20 0.39
ME2 P23368 1/20 0.39
ME1 P48163 1/20 0.39
ME3 Q16798 1/20 0.39
CYP19A1 P11511 1/20 0.39
NQO2 P16083 1/20 0.39
KDM4E B2RXH2 4/20 0.37
ALDH1A1 P00352 2/20 0.37
HPGD P15428 2/20 0.37
RET P07949 2/20 0.36
MEN1 O00255 4/20 0.36
KMT2A Q03164 4/20 0.36
MAPT P10636 3/20 0.36
POLB P06746 1/20 0.36
GAA P10253 1/20 0.36
PKM P14618 1/20 0.36
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
CDK1 P06493 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3182648 0.74 CNR1 (0.48) CNR1CNR2CYP19A1NQO2KDM4E
SCHEMBL8604971 0.72 MTNR1A (0.46) ME2ME1ME3CYP19A1NQO2
SCHEMBL8604209 0.72 EGFR (0.44) ME2ME1ME3KDM4EALDH1A1
SCHEMBL7257608 0.70 RET (0.44) CNR1CNR2CYP19A1NQO2KDM4E
SCHEMBL2430302 0.69 ALDH1A1 (0.46) CNR1CNR2KDM4EALDH1A1MEN1
SCHEMBL6095610 0.68 ALDH1A1 (0.47) CNR2NQO2KDM4EALDH1A1HPGD
SCHEMBL6096141 0.68 HTR2A (0.44) ALDH1A1MEN1KMT2AMAPTGSK3B
SCHEMBL7261266 0.68 ALDH1A1 (0.46) CYP19A1KDM4EALDH1A1HPGDRET
SCHEMBL10839866 0.68 KDM4E (0.65) CNR1CNR2CYP19A1NQO2KDM4E
SCHEMBL7837750 0.66 ALDH1A1 (0.45) CNR1CNR2CYP19A1NQO2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5780496-A Method and compositions for inhibition of adaptor protein/tyrosine kinase interactions SUGEN, INC. (US) 1998-07-14 US claimed
US-5786488-A DEHYDROBROMINATION OF A DIBROMOBENZOQUINONES WITH AT LEAST ONE INDOLES IN A POLAR SOLVENT AND A METAL CARBONATE TO FORM AN ANTITUMOR AGENT SUGEN, INC. (US) 1998-07-28 US disclosed
US-5780496-A Method and compositions for inhibition of adaptor protein/tyrosine kinase interactions SUGEN, INC. (US) 1998-07-14 US disclosed