SCHEMBL8607100

SCHEMBL8607100

Fc1cc(F)cc(P(c2cc(F)cc(F)c2)c2ccc(F)cc2P(c2cc(F)cc(F)c2)c2cc(F)cc(F)c2)c1

nearest known ligand 0.34

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.34
CYP2A6 P11509 1/20 0.34
AHR P35869 1/20 0.30
CA3 P07451 1/20 0.30
CA6 P23280 1/20 0.30
CA5A P35218 1/20 0.30
CA9 Q16790 1/20 0.30
CA14 Q9ULX7 1/20 0.30
CA5B Q9Y2D0 1/20 0.30
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6271249 0.81 CYP1A2 (0.37) CYP1A2CYP2A6CA9
SCHEMBL6250746 0.76 CYP1A2 (0.48) CYP1A2CYP2A6
SCHEMBL1506225 0.74 CA12 (0.42) CA9
SCHEMBL8638150 0.72 CA12 (0.40) CA9
SCHEMBL8675804 0.70 ACHE (0.41) CYP1A2CYP2A6
SCHEMBL6252118 0.68 KMT2A (0.33)
SCHEMBL19921795 0.65 ALDH1A1 (0.46) CYP1A2CYP2A6CA3CA6CA5A
SCHEMBL29716617 0.65 ALDH1A1 (0.46) CYP1A2CYP2A6CA3CA6CA5A
SCHEMBL14369682 0.65 CA3 (0.46) CA3CA6CA5ACA9CA14
SCHEMBL28491054 0.65 CYP3A4 (0.44) CYP1A2CYP2A6CA3CA6CA5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0832087-A1 SYNTHESIS OF AND HYDROFORMYLATION WITH FLUORO-SUBSTITUTED BIDENTATE PHOSPHINE LIGANDS HOECHST CELANESE CORPORATION (US) 1998-04-01 EP claimed
WO-1996038456-A1 SYNTHESIS OF AND HYDROFORMYLATION WITH FLUORO-SUBSTITUTED BIDENTATE PHOSPHINE LIGANDS HOECHST CELANESE CORPORATION (US) 1996-12-05 WO claimed
EP-0832087-A1 SYNTHESIS OF AND HYDROFORMYLATION WITH FLUORO-SUBSTITUTED BIDENTATE PHOSPHINE LIGANDS HOECHST CELANESE CORPORATION (US) 1998-04-01 EP disclosed
US-5616785-A BIS/3,5-DIFLUOROPHENYL/PHOSPHINE OXIDE AND BIS/3,5-DIFLUOROPHENYL/-PHOSPHINOUS ACID; CHEMICAL INTERMEDIATES FOR FLUORO-SUBSTITUTED BIDENTATE PHOSPHINE LIGANDS HOECHST CELANESE CORPORATION (US) 1997-04-01 US disclosed
WO-1996038456-A1 SYNTHESIS OF AND HYDROFORMYLATION WITH FLUORO-SUBSTITUTED BIDENTATE PHOSPHINE LIGANDS HOECHST CELANESE CORPORATION (US) 1996-12-05 WO disclosed
US-5567856-A USING A RHODIUM COMPLEX CATALYST HOECHST CELANESE CORPORATION (US) 1996-10-22 US disclosed