SCHEMBL8610623

SCHEMBL8610623

NN1CCCCC1(Cc1cc(OCC(F)(F)F)ccc1OCC(F)(F)F)c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 2/20 0.47
GRIN2A Q12879 2/20 0.47
GRIN2B Q13224 2/20 0.47
NPSR1 Q6W5P4 1/20 0.36
CYP1A2 P05177 1/20 0.35
CYP2C9 P11712 1/20 0.35
SIGMAR1 Q99720 1/20 0.35
KDM4E B2RXH2 1/20 0.34
SLC6A4 P31645 3/20 0.34
SLC6A2 P23975 1/20 0.34
ALDH1A1 P00352 4/20 0.34
POLB P06746 1/20 0.34
GPR3 P46089 1/20 0.33
ALOX5AP P20292 2/20 0.32
CNR2 P34972 1/20 0.32
TACR1 P25103 2/20 0.32
LMNA P02545 1/20 0.32
TSHR P16473 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8611477 0.89 GRIN1 (0.40) GRIN1GRIN2AGRIN2BSLC6A4SLC6A2
Hydrochloric Acid SCHEMBL8613933 0.88 GRIN1 (0.39) GRIN1GRIN2AGRIN2BSLC6A4SLC6A2
Hydrochloric Acid SCHEMBL8610065 0.85 GRIN1 (0.39) GRIN1GRIN2AGRIN2BSLC6A4SLC6A2
Hydrochloric Acid SCHEMBL8611332 0.85 GRIN1 (0.37) GRIN1GRIN2AGRIN2BNPSR1SLC6A4
Hydrochloric Acid SCHEMBL8614565 0.81 S1PR1 (0.36) GRIN1GRIN2AGRIN2BNPSR1KDM4E
Hydrochloric Acid SCHEMBL8615867 0.78 SLC6A4 (0.37) SIGMAR1SLC6A4SLC6A2ALDH1A1
SCHEMBL7718906 0.75 DRD2 (0.35) GRIN1GRIN2AGRIN2BNPSR1KDM4E
SCHEMBL8706170 0.70 DRD2 (0.34) SLC6A2TACR1
Hydrochloric Acid SCHEMBL8706566 0.69 DRD2 (0.33) SLC6A2TACR1
SCHEMBL8705094 0.69 TACR1 (0.35) NPSR1CYP2C9ALDH1A1TACR1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5773450-A ANTIINFLAMMATORY AGENTS, CENTRAL NERVOUS SYSTEM DISORDERS PFIZER INC. (US) 1998-06-30 US disclosed
US-5744480-A ANTIINFLAMMATORY AGENTS, NERVOUS SYSTEM DISORDERS PFIZER INC. (US) 1998-04-28 US disclosed