SCHEMBL8610947

SCHEMBL8610947

COc1cccc(CNCC(O)CN2CCN(CCCC(c3ccc(F)cc3)c3ccc(F)cc3)CC2)c1OC

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 8/20 0.50
TACR1 P25103 1/20 0.46
MEN1 O00255 3/20 0.45
KMT2A Q03164 3/20 0.45
CYP3A4 P08684 2/20 0.45
CYP2D6 P10635 2/20 0.45
LMNA P02545 2/20 0.45
ADORA3 P0DMS8 2/20 0.45
DRD2 P14416 2/20 0.45
ADRA2B P18089 2/20 0.45
ADRA2C P18825 2/20 0.45
SLC6A2 P23975 2/20 0.45
HTR2A P28223 2/20 0.45
ADRA1A P35348 2/20 0.45
HRH1 P35367 2/20 0.45
DRD3 P35462 2/20 0.45
OPRK1 P41145 2/20 0.45
HTR2B P41595 2/20 0.45
SLC6A3 Q01959 2/20 0.45
GHSR Q92847 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8614292 0.93 KCNH2 (0.52) KCNH2MEN1KMT2ACYP3A4CYP2D6
SCHEMBL9148247 0.84 KCNH2 (0.50) KCNH2TACR1MEN1KMT2ACYP3A4
SCHEMBL8610976 0.82 KCNH2 (0.52) KCNH2MEN1KMT2ACYP3A4CYP2D6
SCHEMBL8611930 0.81 MAPK1 (0.55) KCNH2TACR1MEN1KMT2ACYP3A4
SCHEMBL7751327 0.81 SLC6A3 (0.54) KCNH2MEN1KMT2ACYP3A4CYP2D6
SCHEMBL7754352 0.81 KCNH2 (0.60) KCNH2MEN1KMT2ACYP3A4CYP2D6
SCHEMBL8617368 0.81 KCNH2 (0.52) KCNH2MEN1KMT2ACYP3A4CYP2D6
Hydrochloric Acid SCHEMBL7544797 0.80 SLC6A3 (0.53) MEN1KMT2ACYP3A4CYP2D6ADORA3
SCHEMBL8610943 0.79 KCNH2 (0.51) KCNH2MEN1KMT2ACYP3A4CYP2D6
SCHEMBL8616693 0.78 HTR2A (0.50) KCNH2TACR1MEN1KMT2ACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0549796-B1 DIPHENYLPIPERAZINE DERIVATIVE AND DRUG FOR CIRCULATORY ORGAN CONTAINING THE SAME POLA CHEM IND INC (JP) 1998-04-29 EP disclosed
US-5391552-A Has strong antagonism against calcium with less side effects POLA CHEMICAL INDUSTRIES, INC. (JP) 1995-02-21 US disclosed