SCHEMBL8611031

SCHEMBL8611031

COC(=O)c1cc(S(C)(=O)=O)c(-c2ccccc2)cc1C(C)C

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.48
GABRA1 P14867 1/20 0.44
GABRG2 P18507 1/20 0.44
GABRB3 P28472 1/20 0.44
GABRA3 P34903 1/20 0.44
HPGD P15428 2/20 0.43
KDM4E B2RXH2 1/20 0.43
FGFR1 P11362 1/20 0.43
SRC P12931 1/20 0.43
FGFR2 P21802 1/20 0.43
FGFR4 P22455 1/20 0.43
FGFR3 P22607 1/20 0.43
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA5A P35218 1/20 0.42
CA9 Q16790 1/20 0.42
SLC6A3 Q01959 4/20 0.42
SLC6A4 P31645 3/20 0.42
HTT P42858 1/20 0.42
SLC6A2 P23975 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8610606 0.90 SLC9A1 (0.50) PTGS2KDM4EKMT2AALDH1A1MAPT
SCHEMBL8610875 0.88 CA2 (0.55) PTGS2GABRA1GABRG2GABRB3GABRA3
SCHEMBL8608598 0.87 PTGS2 (0.44) PTGS2GABRA1GABRG2GABRB3GABRA3
SCHEMBL8608047 0.85 PTGS2 (0.52) PTGS2GABRA1GABRG2GABRB3GABRA3
SCHEMBL8608965 0.83 PTGS2 (0.47) PTGS2GABRA1GABRG2GABRB3GABRA3
SCHEMBL8611709 0.80 PTGS2 (0.44) PTGS2GABRA1GABRG2GABRB3GABRA3
SCHEMBL8533240 0.80 SLC9A1 (0.60)
SCHEMBL8608333 0.78 CA2 (0.46) PTGS2KDM4ECA1CA2CA5A
SCHEMBL8607611 0.78 SLC9A1 (0.46) PTGS2KDM4EALDH1A1MAPT
SCHEMBL8608602 0.78 PTGS2 (0.43) PTGS2GABRA1GABRG2GABRB3GABRA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5807896-A Arylbenzoylguanidines MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTING (DE) 1998-09-15 US disclosed