SCHEMBL8637503

SCHEMBL8637503

CCOc1ccccc1N1CCN(CC(O)COc2ccccc2NC(=O)CC)CC1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 7/20 0.60
ADRA1B P35368 3/20 0.54
ALDH1A1 P00352 3/20 0.53
KDM4E B2RXH2 2/20 0.53
USP2 O75604 2/20 0.53
TSHR P16473 2/20 0.53
HSD17B10 Q99714 1/20 0.53
MAPT P10636 4/20 0.53
LMNA P02545 3/20 0.52
MEN1 O00255 3/20 0.52
KMT2A Q03164 3/20 0.52
MAPK1 P28482 2/20 0.52
TDP1 Q9NUW8 2/20 0.52
NR1I2 O75469 1/20 0.52
NR3C1 P04150 1/20 0.52
ADRB1 P08588 1/20 0.52
HTR1A P08908 1/20 0.52
ADRA2A P08913 1/20 0.52
DRD2 P14416 1/20 0.52
ADRA2B P18089 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8615289 0.92 MAPT (0.63) ABCB1ADRA1BALDH1A1KDM4EUSP2
SCHEMBL8615117 0.82 MAPT (0.66) ABCB1ADRA1BALDH1A1KDM4EUSP2
SCHEMBL8609331 0.82 MAPT (0.66) ABCB1ADRA1BALDH1A1KDM4EUSP2
SCHEMBL4753120 0.81 LMNA (0.74) ABCB1ADRA1BALDH1A1KDM4EUSP2
SCHEMBL8611715 0.80 HSP90AB1 (0.58) ABCB1ADRA1BALDH1A1KDM4EUSP2
SCHEMBL8645443 0.80 ABCB1 (0.73) ABCB1
SCHEMBL8609924 0.80 MAPT (0.62) ABCB1ADRA1BALDH1A1KDM4EUSP2
SCHEMBL11808577 0.77 CACNA1G (0.66) ABCB1ALDH1A1KDM4EUSP2TSHR
SCHEMBL8613687 0.77 HSP90AB1 (0.55) ABCB1KCNH2
SCHEMBL31448071 0.77 LMNA (0.73) ABCB1ALDH1A1USP2MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0833639-A1 PHENOXY PIPERAZINE DERIVATIVES FOR TREATING DISORDERS OF THE DOPAMINE SYSTEM F. HOFFMANN-LA ROCHE AG (CH) 1998-04-08 EP disclosed
US-5614526-A IN TREATING DISORDERS OF THE DOPAMINE SYSTEM HOFFMANN-LA ROCHE INC. (US) 1997-03-25 US disclosed
WO-1996041630-A1 PHENOXY PIPERAZINE DERIVATIVES FOR TREATING DISORDERS OF THE DOPAMINE SYSTEM F. HOFFMANN-LA ROCHE AG (CH) 1996-12-27 WO disclosed