SCHEMBL8612679

SCHEMBL8612679

CC(=O)Nc1ccc2c(NC(=N)NC=O)cc(-c3ccccc3)nc2c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 1/20 0.55
ABCC1 P33527 1/20 0.55
ABCG2 Q9UNQ0 1/20 0.55
KMT2A Q03164 6/20 0.51
MEN1 O00255 5/20 0.51
ALDH1A1 P00352 6/20 0.49
TP53 P04637 1/20 0.49
CYP1A2 P05177 1/20 0.49
HSD17B10 Q99714 1/20 0.49
KDM4E B2RXH2 6/20 0.49
MAPT P10636 3/20 0.49
HPGD P15428 2/20 0.49
PDE10A Q9Y233 2/20 0.49
NPSR1 Q6W5P4 1/20 0.49
RXFP1 Q9HBX9 1/20 0.49
CYP2C19 P33261 1/20 0.49
MOK Q9UQ07 6/20 0.48
NPC1 O15118 2/20 0.45
RAB9A P51151 2/20 0.45
POLB P06746 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8617766 0.93 ABCB1 (0.54) ABCB1ABCC1ABCG2KMT2AMEN1
SCHEMBL8619415 0.90 ABCB1 (0.47) ABCB1ABCC1ABCG2KMT2AMEN1
SCHEMBL8615149 0.87 ALDH1A1 (0.49) ABCB1ABCC1ABCG2KMT2AMEN1
SCHEMBL8613684 0.87 NPC1 (0.42) ABCB1ABCC1ABCG2KMT2AMEN1
SCHEMBL8617739 0.86 ALDH1A1 (0.47) ABCB1ABCC1ABCG2ALDH1A1HSD17B10
SCHEMBL8617753 0.85 ACP1 (0.51) ABCB1ABCC1ABCG2KMT2AMEN1
SCHEMBL8615210 0.84 TACR3 (0.44) ABCB1ABCC1ABCG2KMT2AMEN1
SCHEMBL8619389 0.84 TACR3 (0.41) ABCB1ABCC1ABCG2ALDH1A1HSD17B10
SCHEMBL8615938 0.84 TACR3 (0.41) ABCB1ABCC1ABCG2KMT2ATACR3
SCHEMBL8618234 0.84 RXFP1 (0.44) ABCB1ABCC1ABCG2ALDH1A1RXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed