SCHEMBL8613684

SCHEMBL8613684

CC(=O)Nc1ccc2c(NC(=N)NC=O)cc(-c3ccccc3C)nc2c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 7/20 0.42
KMT2A Q03164 7/20 0.42
KDM4E B2RXH2 6/20 0.42
RAB9A P51151 6/20 0.42
MEN1 O00255 6/20 0.42
MAPT P10636 5/20 0.42
PABPC1 P11940 1/20 0.42
ABCB1 P08183 1/20 0.41
ABCC1 P33527 1/20 0.41
ABCG2 Q9UNQ0 1/20 0.41
GLA P06280 1/20 0.38
TNNI3 P19429 1/20 0.38
TNNT2 P45379 1/20 0.38
TNNC1 P63316 1/20 0.38
RUNX1 Q01196 1/20 0.38
CBFB Q13951 1/20 0.38
ALDH1A1 P00352 4/20 0.38
TP53 P04637 3/20 0.38
SMN1; SMN2 Q16637 3/20 0.38
HSD17B10 Q99714 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8613752 0.92 KMT2A (0.42) NPC1KMT2AKDM4ERAB9AMEN1
SCHEMBL8617771 0.87 ALDH1A1 (0.40) NPC1KDM4ERAB9AMAPTGLA
SCHEMBL8620107 0.87 HTT (0.37) KMT2AKDM4EMEN1MAPTRUNX1
SCHEMBL8612679 0.87 ABCB1 (0.55) NPC1KMT2AKDM4ERAB9AMEN1
SCHEMBL8620892 0.86 HTT (0.47) KMT2AKDM4ERAB9AMEN1MAPT
SCHEMBL8619346 0.84 TACR3 (0.46) KDM4EMAPTGLAALDH1A1TP53
SCHEMBL8615234 0.83 HTT (0.38) NPC1KMT2AKDM4ERAB9AMEN1
SCHEMBL8618049 0.82 KDM4E (0.41) NPC1KMT2AKDM4ERAB9AMEN1
SCHEMBL8617546 0.82 ALDH1A1 (0.41) KMT2AKDM4EMEN1MAPTALDH1A1
SCHEMBL8613388 0.82 SMN1; SMN2 (0.39) NPC1KMT2AKDM4ERAB9AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed