SCHEMBL8613889

SCHEMBL8613889

N=C(N)NC(=O)c1cc(-c2ccccc2)nc2c(NC(=O)C3CCCC3)cccc12

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 9/20 0.50
ADORA2A P29274 6/20 0.50
ADORA3 P0DMS8 5/20 0.50
CYP2C9 P11712 2/20 0.43
ALDH1A1 P00352 3/20 0.42
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
GFER P55789 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
ALOX12 P18054 1/20 0.42
CYP2C19 P33261 1/20 0.42
KDM4E B2RXH2 1/20 0.41
HPGD P15428 1/20 0.41
KCNH2 Q12809 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8618987 0.84 KMT2A (0.51) ADORA1ADORA3CYP2C9ALDH1A1MEN1
SCHEMBL8613213 0.81 KMT2A (0.47) ADORA1ADORA3CYP2C9ALDH1A1MEN1
SCHEMBL8618761 0.80 MEN1 (0.56) CYP2C9ALDH1A1MEN1KMT2ACYP1A2
SCHEMBL8619721 0.79 MEN1 (0.45) CYP2C9ALDH1A1MEN1KMT2AGFER
SCHEMBL8615990 0.78 CCR6 (0.57) CYP2C9ALDH1A1MEN1KMT2AGFER
SCHEMBL8616695 0.78 MEN1 (0.46) CYP2C9ALDH1A1MEN1KMT2AGFER
SCHEMBL8620933 0.78 ADORA1 (0.47) ADORA1ADORA2AADORA3CYP2C9ALDH1A1
SCHEMBL8614378 0.78 MEN1 (0.44) CYP2C9ALDH1A1MEN1KMT2AGFER
SCHEMBL8619899 0.78 MEN1 (0.46) CYP2C9ALDH1A1MEN1KMT2AGFER
SCHEMBL8613481 0.78 KDM4E (0.56) CYP2C9ALDH1A1MEN1KMT2ACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed