SCHEMBL8618987

SCHEMBL8618987

CC(=O)Nc1cccc2c(C(=O)NC(=N)N)cc(-c3ccccc3)nc12

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 8/20 0.51
MEN1 O00255 7/20 0.51
ALDH1A1 P00352 5/20 0.48
CYP3A4 P08684 3/20 0.48
CYP2C9 P11712 2/20 0.48
CYP1A2 P05177 2/20 0.48
ALOX12 P18054 2/20 0.48
CYP2C19 P33261 2/20 0.48
GFER P55789 1/20 0.47
PTGER4 P35408 1/20 0.46
KDM4E B2RXH2 3/20 0.45
KCNH2 Q12809 2/20 0.45
ABCB1 P08183 1/20 0.45
ABCC1 P33527 1/20 0.45
ABCG2 Q9UNQ0 1/20 0.45
HPGD P15428 1/20 0.45
PDE10A Q9Y233 2/20 0.45
ADORA3 P0DMS8 1/20 0.44
ADORA1 P30542 1/20 0.44
POLB P06746 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8613213 0.96 KMT2A (0.47) KMT2AMEN1ALDH1A1CYP3A4CYP2C9
SCHEMBL8617543 0.87 MEN1 (0.46) KMT2AMEN1ALDH1A1CYP3A4CYP2C9
SCHEMBL8619721 0.85 MEN1 (0.45) KMT2AMEN1ALDH1A1CYP3A4CYP2C9
SCHEMBL8614378 0.85 MEN1 (0.44) KMT2AMEN1ALDH1A1CYP3A4CYP2C9
SCHEMBL8620933 0.85 ADORA1 (0.47) KMT2AMEN1ALDH1A1CYP3A4CYP2C9
SCHEMBL8613481 0.84 KDM4E (0.56) KMT2AMEN1ALDH1A1CYP3A4CYP2C9
SCHEMBL8613889 0.84 ADORA1 (0.50) KMT2AMEN1ALDH1A1CYP3A4CYP2C9
SCHEMBL8618698 0.84 PDE10A (0.62) KMT2AMEN1ALDH1A1CYP1A2GFER
SCHEMBL8615990 0.83 CCR6 (0.57) KMT2AMEN1ALDH1A1CYP3A4CYP2C9
SCHEMBL8616695 0.83 MEN1 (0.46) KMT2AMEN1ALDH1A1CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed