SCHEMBL8617812

SCHEMBL8617812

N=C(NC=O)Nc1cc(-c2ccccc2)nc2ccc(Cl)cc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.46
CYP2C9 P11712 3/20 0.44
PTGES O14684 2/20 0.44
ALDH1A1 P00352 1/20 0.44
ALOX5 P09917 1/20 0.44
HPGD P15428 1/20 0.44
CASP7 P55210 1/20 0.44
HIF1A Q16665 1/20 0.44
HSD17B10 Q99714 1/20 0.44
DHODH Q02127 3/20 0.43
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA9 Q16790 1/20 0.43
AURKA O14965 1/20 0.43
AURKB Q96GD4 1/20 0.43
FABP3 P05413 1/20 0.41
FABP4 P15090 1/20 0.41
ACACA Q13085 1/20 0.41
MAPT P10636 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8619389 0.92 TACR3 (0.41) MAPK1CYP2C9PTGESALDH1A1ALOX5
SCHEMBL8615684 0.87 ESR1 (0.43) MEN1KMT2AACP1
SCHEMBL8617753 0.87 ACP1 (0.51) MEN1KMT2AKDM4ELMNAACP1
SCHEMBL8614079 0.86 ACP1 (0.52) ALDH1A1CA12CA1CA2CA9
SCHEMBL8613853 0.86 ALDH1A1 (0.52) MAPK1CYP2C9ALDH1A1HPGDHSD17B10
SCHEMBL8615496 0.86 DHODH (0.50) ALDH1A1DHODHMEN1KMT2APLA2G2A
SCHEMBL8617521 0.86 TLR9 (0.41) ALDH1A1HPGDMAPTMEN1KMT2A
SCHEMBL8614838 0.86 MEN1 (0.40) CYP2C9MEN1KMT2AKDM4ELMNA
SCHEMBL8613674 0.83 TRPV1 (0.43) CYP2C9ALDH1A1HPGDMAPTMEN1
SCHEMBL8620945 0.83 NQO2 (0.56) ALDH1A1CA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed