SCHEMBL8615786

SCHEMBL8615786

CC(Cc1ccc(Cl)cc1)NCc1ccc(-c2ccccc2)cc1

nearest known ligand 0.69

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 5/20 0.69
LMNA P02545 2/20 0.56
CYP1A2 P05177 4/20 0.52
CYP2D6 P10635 3/20 0.52
CYP2C19 P33261 1/20 0.52
MAPK1 P28482 2/20 0.50
ALDH1A1 P00352 2/20 0.50
HTT P42858 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
AKT1 P31749 1/20 0.50
POLB P06746 1/20 0.48
TDP1 Q9NUW8 1/20 0.47
KCNH2 Q12809 1/20 0.47
TMEM97 Q5BJF2 1/20 0.47
PPARG P37231 1/20 0.47
PPARA Q07869 1/20 0.47
CYP3A4 P08684 1/20 0.46
TSHR P16473 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8091283 0.93 SIGMAR1 (0.79) SIGMAR1LMNACYP1A2CYP2D6CYP2C19
N-Benzylamphetamine SCHEMBL2451256 0.82 SIGMAR1 (1.00) SIGMAR1LMNACYP1A2CYP2D6MAPK1
N-Benzylamphetamine SCHEMBL2795222 0.82 SIGMAR1 (1.00) SIGMAR1LMNACYP1A2CYP2D6MAPK1
N-Benzylamphetamine SCHEMBL2798189 0.82 SIGMAR1 (1.00) SIGMAR1LMNACYP1A2CYP2D6MAPK1
N-Benzylamphetamine SCHEMBL8085021 0.81 SIGMAR1 (0.96) SIGMAR1LMNACYP1A2CYP2D6MAPK1
SCHEMBL8587928 0.80 DPP7 (0.47) SIGMAR1LMNACYP1A2CYP2D6CYP2C19
SCHEMBL24997843 0.80 SIGMAR1 (0.79) SIGMAR1LMNACYP1A2CYP2D6MAPK1
SCHEMBL606189 0.80 SIGMAR1 (0.85) SIGMAR1LMNACYP1A2CYP2D6MAPK1
SCHEMBL12377261 0.79 CYP1A2 (0.49) LMNACYP1A2CYP2D6CYP2C19MAPK1
SCHEMBL608555 0.78 SIGMAR1 (0.82) SIGMAR1LMNACYP1A2CYP2D6MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998052890-A1 3-ARYLPROPYLAMINO NEUROPEPTIDE Y RECEPTOR ANTAGONISTS ELI LILLY AND COMPANY (US) 1998-11-26 WO disclosed