SCHEMBL8615841

SCHEMBL8615841

COc1ccc(C)c2nc(-c3ccccc3C)cc(C(=O)NC(=N)N)c12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 1/20 0.39
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA9 Q16790 1/20 0.39
KMT2A Q03164 5/20 0.39
MEN1 O00255 3/20 0.39
ALDH1A1 P00352 4/20 0.38
HPGD P15428 4/20 0.38
KDM4E B2RXH2 4/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
TP53 P04637 1/20 0.37
MAPT P10636 3/20 0.37
HTT P42858 3/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
ADORA2A P29274 1/20 0.37
ADORA1 P30542 1/20 0.37
GPR55 Q9Y2T6 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8619166 0.95 TACR3 (0.40) TACR3CA12CA1CA2CA9
SCHEMBL8620849 0.92 TACR3 (0.39) TACR3CA12CA1CA2CA9
SCHEMBL8617698 0.91 CA2 (0.41) TACR3CA12CA1CA2CA9
SCHEMBL8614893 0.91 CA2 (0.39) TACR3CA12CA1CA2CA9
SCHEMBL8616039 0.91 TACR3 (0.38) TACR3CA12CA1CA2CA9
SCHEMBL8618478 0.88 THRB (0.39) TACR3CA12CA1CA2CA9
SCHEMBL8614889 0.87 CA2 (0.39) TACR3CA12CA1CA2CA9
SCHEMBL8617514 0.87 TACR3 (0.38) TACR3CA12CA1CA2CA9
SCHEMBL8618641 0.87 CCNT1 (0.38) TACR3CA12CA1CA2CA9
SCHEMBL8615515 0.87 KMT2A (0.41) TACR3CA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed