SCHEMBL8618641

SCHEMBL8618641

COc1ccc(F)c2c(C(=O)NC(=N)N)cc(-c3ccccc3C)nc12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNT1 O60563 1/20 0.38
CDK9 P50750 1/20 0.38
TACR3 P29371 1/20 0.38
ALDH1A1 P00352 2/20 0.37
HTT P42858 2/20 0.37
MAPT P10636 2/20 0.37
HCRTR1 O43613 1/20 0.37
HCRTR2 O43614 1/20 0.37
HPGD P15428 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
GPR55 Q9Y2T6 1/20 0.37
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA9 Q16790 1/20 0.37
CTSA P10619 3/20 0.37
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
ADORA2A P29274 2/20 0.35
ADORA1 P30542 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8619166 0.92 TACR3 (0.40) TACR3ALDH1A1HTTMAPTHPGD
SCHEMBL8620849 0.91 TACR3 (0.39) TACR3ALDH1A1HTTMAPTHPGD
SCHEMBL8617698 0.89 CA2 (0.41) TACR3ALDH1A1HTTMAPTHPGD
SCHEMBL8615515 0.89 KMT2A (0.41) TACR3ALDH1A1HTTMAPTHPGD
SCHEMBL8614889 0.89 CA2 (0.39) TACR3ALDH1A1HTTMAPTHPGD
SCHEMBL8617514 0.89 TACR3 (0.38) TACR3ALDH1A1HTTMAPTHPGD
SCHEMBL8615841 0.87 TACR3 (0.39) TACR3ALDH1A1HTTMAPTHCRTR2
SCHEMBL8616639 0.85 THRB (0.39) TACR3ALDH1A1HTTMAPTHPGD
SCHEMBL8616039 0.85 TACR3 (0.38) TACR3ALDH1A1HTTMAPTHPGD
SCHEMBL8614893 0.85 CA2 (0.39) TACR3ALDH1A1HTTMAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed