SCHEMBL8616670

SCHEMBL8616670

COc1ccc2nc(-c3ccccc3C)cc(C(=O)NC(=N)N)c2c1

nearest known ligand 0.65

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CA9 Q16790 9/20 0.65
CA2 P00918 8/20 0.65
CA12 O43570 7/20 0.65
CA1 P00915 6/20 0.65
PLA2G2A P14555 2/20 0.53
TACR3 P29371 3/20 0.50
HTT P42858 2/20 0.47
ALDH1A1 P00352 2/20 0.47
HPGD P15428 2/20 0.47
MAPT P10636 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
GPR55 Q9Y2T6 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C9 P11712 1/20 0.47
PLA2G10 O15496 1/20 0.47
KDM4E B2RXH2 2/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
POLB P06746 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8619345 0.92 CA2 (0.55) CA9CA2CA12CA1TACR3
SCHEMBL8619081 0.90 CA2 (0.56) CA9CA2CA12CA1PLA2G2A
SCHEMBL8615492 0.89 CA2 (0.53) CA9CA2CA12CA1TACR3
SCHEMBL8620936 0.87 PLA2G2A (0.69) CA9CA2CA12CA1PLA2G2A
SCHEMBL8618109 0.87 CA2 (0.51) CA9CA2CA12CA1PLA2G2A
SCHEMBL8617885 0.87 CA2 (0.49) CA9CA2CA12CA1TACR3
SCHEMBL8614945 0.86 ALDH1A1 (0.51) CA9CA2CA12CA1TACR3
SCHEMBL8620889 0.86 HTT (0.61) TACR3HTTALDH1A1HPGDMAPT
SCHEMBL8617712 0.86 CA2 (0.50) CA9CA2CA12CA1TACR3
SCHEMBL8614152 0.86 CA9 (0.50) CA9CA2CA12CA1PLA2G2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed