SCHEMBL8617124

SCHEMBL8617124

CCCCCOc1cccc2nc(-c3ccccc3C)cc(NC(=N)NC=O)c12

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR8 Q9NR97 3/20 0.36
KMT2A Q03164 2/20 0.34
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HPGD P15428 1/20 0.34
DNMT1 P26358 1/20 0.34
EHMT2 Q96KQ7 1/20 0.34
NCF1 P14598 1/20 0.33
PTPN11 Q06124 1/20 0.33
TACR3 P29371 1/20 0.33
CNR2 P34972 3/20 0.33
ACP1 P24666 1/20 0.33
TP53 P04637 1/20 0.33
PTGER1 P34995 1/20 0.33
PTPN1 P18031 1/20 0.33
HTT P42858 1/20 0.33
CSNK1A1 P48729 1/20 0.32
CSNK1D P48730 1/20 0.32
PRKCD Q05655 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8618522 0.95 ABL1 (0.36) TLR8KMT2AKDM4EMEN1ALDH1A1
SCHEMBL8615341 0.91 MEN1 (0.39) KMT2AKDM4EMEN1ALDH1A1HPGD
SCHEMBL8618132 0.89 DNMT1 (0.36) KMT2AKDM4EMEN1ALDH1A1HPGD
SCHEMBL8613232 0.88 TACR3 (0.36) KMT2AKDM4EMEN1ALDH1A1HPGD
SCHEMBL8617965 0.88 NCF1 (0.33) KMT2AKDM4EMEN1ALDH1A1HPGD
SCHEMBL8614832 0.87 MEN1 (0.33) KMT2AKDM4EMEN1ALDH1A1HPGD
SCHEMBL8617704 0.86 KDM4E (0.33) KMT2AKDM4EMEN1ALDH1A1HPGD
SCHEMBL8619913 0.86 TGFBR1 (0.39) KMT2AKDM4EMEN1ALDH1A1HPGD
SCHEMBL8617850 0.86 S1PR5 (0.37) HPGDCNR2
SCHEMBL8620877 0.84 HTT (0.39) KMT2AKDM4EMEN1ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed