SCHEMBL8617850

SCHEMBL8617850

CCCCCOc1cccc2c(NC(=N)NC=O)cc(-c3ccccc3C)nc12

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
S1PR5 Q9H228 2/20 0.37
HPGD P15428 1/20 0.36
MAPK1 P28482 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
GAA P10253 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
SLC6A4 P31645 1/20 0.36
CNR1 P21554 2/20 0.36
CNR2 P34972 2/20 0.36
CYP2C9 P11712 1/20 0.36
HTR1B P28222 1/20 0.35
MCL1 Q07820 2/20 0.35
S1PR2 O95136 1/20 0.35
S1PR1 P21453 1/20 0.35
S1PR3 Q99500 1/20 0.35
LPAR2 Q9HBW0 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8617193 0.97 GAA (0.39) HPGDMAPK1NPSR1GAATDP1
SCHEMBL8614073 0.97 S1PR5 (0.37) S1PR5HPGDMAPK1NPSR1GAA
SCHEMBL8617403 0.91 KMT2A (0.41) L3MBTL1
SCHEMBL8615146 0.89 ALDH1A1 (0.41) HPGDNPSR1GAAL3MBTL1SLC6A4
SCHEMBL8617986 0.86 KDM4E (0.32) HPGDL3MBTL1
SCHEMBL8613400 0.86 GFER (0.41) HPGDGAATDP1
SCHEMBL8617124 0.86 TLR8 (0.36) HPGDCNR2
SCHEMBL8620384 0.84 MCHR1 (0.36) HPGDL3MBTL1SLC6A4
SCHEMBL8620017 0.84 DHODH (0.37) HPGDNPSR1SLC6A4
SCHEMBL8618902 0.84 TACR3 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed