SCHEMBL8617375

SCHEMBL8617375

CCCCN(CC)c1cc(C)nc2c1c(C)c(C)n2-c1c(C)cc(C)cc1C

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CRHR1 P34998 14/20 1.00
TDP1 Q9NUW8 2/20 0.69
FPR3 P25089 2/20 0.47
TSPO P30536 2/20 0.47
TMEM97 Q5BJF2 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8619340 0.88 CRHR1 (0.79) CRHR1TDP1
SCHEMBL7215696 0.82 CRHR1 (0.69) CRHR1TDP1FPR3TSPOTMEM97
SCHEMBL7222252 0.82 CRHR1 (0.69) CRHR1TDP1FPR3TSPOTMEM97
SCHEMBL5599498 0.82 CRHR1 (0.72) CRHR1TDP1FPR3TSPOTMEM97
Antalarmin SCHEMBL466243 0.82 CRHR1 (1.00) CRHR1TDP1FPR3TSPOTMEM97
Antalarmin SCHEMBL29832078 0.82 CRHR1 (1.00) CRHR1TDP1FPR3TSPOTMEM97
Antalarmin SCHEMBL25395568 0.81 CRHR1 (0.98) CRHR1TDP1FPR3TSPOTMEM97
Antalarmin SCHEMBL29601552 0.81 CRHR1 (0.98) CRHR1TDP1FPR3TSPOTMEM97
SCHEMBL8621371 0.81 CRHR1 (0.67) CRHR1TDP1
SCHEMBL6295510 0.75 CRHR1 (0.69) CRHR1FPR3TSPOTMEM97

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998045295-A1 CERTAIN PYRROLOPYRIDINE DERIVATIVES; NOVEL CRF1 SPECIFIC LIGANDS NEUROGEN CORPORATION (US) 1998-10-15 WO claimed
WO-1998045295-A1 CERTAIN PYRROLOPYRIDINE DERIVATIVES; NOVEL CRF1 SPECIFIC LIGANDS NEUROGEN CORPORATION (US) 1998-10-15 WO disclosed