SCHEMBL8617666

SCHEMBL8617666

CCC(C)OP(=O)(O)CNc1c(N)ccc2c(S(N)(=O)=O)cccc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 2/20 0.39
CA2 P00918 3/20 0.34
AURKA O14965 1/20 0.33
AURKB Q96GD4 1/20 0.33
KDM4E B2RXH2 1/20 0.32
MEN1 O00255 1/20 0.32
USP2 O75604 1/20 0.32
ALDH1A1 P00352 1/20 0.32
LMNA P02545 1/20 0.32
TSHR P16473 1/20 0.32
MAPK1 P28482 1/20 0.32
HTT P42858 1/20 0.32
KMT2A Q03164 1/20 0.32
CA1 P00915 2/20 0.32
CA9 Q16790 1/20 0.32
NSD2 O96028 6/20 0.32
NR4A1 P22736 1/20 0.32
LDHA P00338 1/20 0.32
TTR P02766 1/20 0.31
CYP1A2 P05177 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8619769 0.87 CDK2 (0.36) CDK2CA2KDM4EMEN1ALDH1A1
SCHEMBL8622828 0.84 CDK2 (0.38) CDK2CA2AURKAAURKBKDM4E
SCHEMBL8623611 0.84 CDK2 (0.38) CDK2CA2KDM4EMEN1USP2
SCHEMBL8617963 0.81 MAPT (0.39) CA2KDM4EMEN1ALDH1A1KMT2A
SCHEMBL8619789 0.81 CDK2 (0.35) CDK2CA2KDM4EMEN1USP2
SCHEMBL8623637 0.79 MAPT (0.40) CA2KDM4EMEN1ALDH1A1LMNA
SCHEMBL8617656 0.78 CDK2 (0.38) CDK2CA2KDM4ELMNAMAPK1
SCHEMBL8616429 0.74 MAPT (0.42) KDM4EMEN1ALDH1A1LMNAMAPK1
SCHEMBL9037282 0.74 CA2 (0.34) CDK2CA2CA1CA9
SCHEMBL8622818 0.73 CA2 (0.38) CDK2CA2KDM4EALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5710138-A Benzo f!quinoxalinedione derivatives, their production and use in pharmaceutical agents SCHERING AKTIENGESELLSCHAFT (DE) 1998-01-20 US disclosed