SCHEMBL8618326

SCHEMBL8618326

C[C@]12CC[C@@H]3c4ccc(OC(=O)c5ccccc5)cc4CC[C@H]3[C@@H]1C[C@@H](O)[C@@H]2OC(=O)COC(=O)CCCc1ccc(N(CCCl)CCCl)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 4/20 0.53
ADORA3 P0DMS8 3/20 0.53
SMN1; SMN2 Q16637 3/20 0.53
ATM Q13315 3/20 0.53
LMNA P02545 2/20 0.53
KMT2A Q03164 2/20 0.53
NR3C1 P04150 1/20 0.53
SHBG P04278 1/20 0.53
FYN P06241 1/20 0.53
ADRA2C P18825 1/20 0.53
SLC6A2 P23975 1/20 0.53
SLC6A4 P31645 1/20 0.53
HTR2B P41595 1/20 0.53
HTT P42858 1/20 0.53
RECQL P46063 1/20 0.48
BLM P54132 1/20 0.48
CYP3A4 P08684 3/20 0.47
MAPT P10636 3/20 0.45
USP2 O75604 1/20 0.45
MAPK1 P28482 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8656096 0.92 ESR1 (0.49) ESR1ADORA3SMN1; SMN2ATMLMNA
Atrimustine SCHEMBL10580413 0.90 LMNA (0.56) ESR1ADORA3SMN1; SMN2ATMLMNA
Atrimustine SCHEMBL29359877 0.90 LMNA (0.56) ESR1ADORA3SMN1; SMN2ATMLMNA
Atrimustine SCHEMBL8659 0.90 LMNA (0.56) ESR1ADORA3SMN1; SMN2ATMLMNA
SCHEMBL8836343 0.85 LMNA (0.58) ESR1ADORA3SMN1; SMN2ATMLMNA
SCHEMBL9319675 0.81 LMNA (0.56) ESR1ADORA3SMN1; SMN2ATMLMNA
SCHEMBL8835854 0.81 LMNA (0.56) ESR1ADORA3SMN1; SMN2ATMLMNA
SCHEMBL8615788 0.80 KMT2A (0.44) ESR1ADORA3SMN1; SMN2ATMLMNA
SCHEMBL8621073 0.80 MAPT (0.46) ESR1ADORA3SMN1; SMN2ATMLMNA
SCHEMBL8619796 0.80 LMNA (0.69) ESR1ADORA3SMN1; SMN2ATMLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0573977-B1 Novel estradiol derivative-chlorambucil conjugate, process for preparing the same, and pharmaceutical composition KUREHA CHEMICAL IND CO LTD (JP) 1998-05-13 EP disclosed
EP-0573977-A2 Novel estradiol derivative-chlorambucil conjugate, process for preparing the same, and pharmaceutical composition KUREHA CHEMICAL INDUSTRY CO., LTD. (JP) 1993-12-15 EP disclosed