SCHEMBL8618698

SCHEMBL8618698

CC(=O)Nc1cccc2c(C(=O)O)cc(-c3ccccc3)nc12

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 3/20 0.62
KDM4E B2RXH2 4/20 0.60
KMT2A Q03164 3/20 0.60
LMNA P02545 2/20 0.56
SMN1; SMN2 Q16637 1/20 0.56
PPARA Q07869 1/20 0.55
MEN1 O00255 2/20 0.54
GFER P55789 1/20 0.54
HTT P42858 1/20 0.54
ALDH1A1 P00352 2/20 0.54
HSD17B10 Q99714 2/20 0.54
TP53 P04637 1/20 0.54
CYP1A2 P05177 1/20 0.54
DHODH Q02127 1/20 0.53
ADORA3 P0DMS8 1/20 0.52
ADORA1 P30542 1/20 0.52
ABCB1 P08183 1/20 0.52
ABCC1 P33527 1/20 0.52
ABCG2 Q9UNQ0 1/20 0.52
AURKA O14965 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8617075 0.85 CCR6 (0.71) PDE10AKDM4EKMT2ASMN1; SMN2MEN1
SCHEMBL8618987 0.84 KMT2A (0.51) PDE10AKDM4EKMT2AMEN1GFER
SCHEMBL8613469 0.82 PDE10A (0.59) PDE10AKDM4EKMT2ALMNASMN1; SMN2
SCHEMBL8613213 0.81 KMT2A (0.47) PDE10AKDM4EKMT2AMEN1GFER
SCHEMBL11810641 0.81 PDE10A (0.70) PDE10AKDM4ELMNASMN1; SMN2PPARA
SCHEMBL6429299 0.80 KDM4E (0.80) PDE10AKDM4ELMNASMN1; SMN2PPARA
SCHEMBL19475364 0.78 KMT2A (0.69) PDE10AKDM4EKMT2APPARAMEN1
SCHEMBL13958056 0.78 CCR6 (0.68) PDE10AKDM4ELMNASMN1; SMN2PPARA
SCHEMBL1901803 0.78 KDM4E (0.77) PDE10AKDM4EKMT2ALMNASMN1; SMN2
SCHEMBL8618998 0.77 ABCB1 (0.47) PDE10AKDM4EKMT2ASMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed