SCHEMBL8619083

SCHEMBL8619083

Cc1ccccc1-c1cc(NC(=N)NC=O)c2cc(OC(C)C)ccc2n1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 4/20 0.44
CA9 Q16790 4/20 0.44
CA12 O43570 3/20 0.44
CA1 P00915 2/20 0.44
TACR3 P29371 1/20 0.39
HTT P42858 4/20 0.38
ALDH1A1 P00352 5/20 0.38
HPGD P15428 5/20 0.38
MAPT P10636 4/20 0.38
MEN1 O00255 4/20 0.38
KMT2A Q03164 4/20 0.38
SMN1; SMN2 Q16637 4/20 0.38
KDM4E B2RXH2 4/20 0.38
POLB P06746 2/20 0.38
LMNA P02545 2/20 0.38
GALR3 O60755 1/20 0.38
CACNA1B Q00975 1/20 0.38
APBA1 Q02410 1/20 0.38
GPR55 Q9Y2T6 1/20 0.37
ACP1 P24666 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8618115 0.91 CA2 (0.40) CA2CA9CA12CA1TACR3
SCHEMBL8616673 0.89 CA2 (0.50) CA2CA9CA12CA1TACR3
SCHEMBL8615494 0.87 SMN1; SMN2 (0.42) CA2CA9CA12CA1TACR3
SCHEMBL8618941 0.87 CA2 (0.38) CA2CA9CA12CA1TACR3
SCHEMBL8618215 0.86 CA2 (0.37) CA2CA9CA12CA1TACR3
SCHEMBL8614156 0.84 CA2 (0.39) CA2CA9CA12CA1TACR3
SCHEMBL8614948 0.84 HTT (0.39) CA2CA9CA12CA1TACR3
SCHEMBL8620892 0.84 HTT (0.47) TACR3HTTALDH1A1HPGDMAPT
SCHEMBL8617721 0.84 CA2 (0.38) CA2CA9CA12CA1TACR3
SCHEMBL8614075 0.84 CA2 (0.38) CA2CA9CA12CA1TACR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed