SCHEMBL8614948

SCHEMBL8614948

Cc1ccccc1-c1cc(NC(=N)NC=O)c2cc(O)ccc2n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.39
ALDH1A1 P00352 6/20 0.39
HPGD P15428 5/20 0.39
KDM4E B2RXH2 4/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
POLB P06746 1/20 0.38
MAPT P10636 2/20 0.36
TACR3 P29371 1/20 0.36
ALOX12 P18054 1/20 0.36
MAPK10 P53779 1/20 0.36
ATM Q13315 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
GPR55 Q9Y2T6 1/20 0.36
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA9 Q16790 1/20 0.36
CYP1A2 P05177 2/20 0.36
CYP2C9 P11712 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8620107 0.92 HTT (0.37) HTTALDH1A1HPGDKDM4EMEN1
SCHEMBL8620892 0.89 HTT (0.47) HTTALDH1A1HPGDKDM4EMEN1
SCHEMBL8615234 0.88 HTT (0.38) HTTALDH1A1HPGDKDM4EMEN1
SCHEMBL8616673 0.87 CA2 (0.50) KDM4EMEN1KMT2AMAPTTACR3
SCHEMBL8613752 0.87 KMT2A (0.42) HTTALDH1A1HPGDKDM4EMEN1
SCHEMBL8615684 0.85 ESR1 (0.43) MEN1KMT2APOLBTACR3CYP3A4
SCHEMBL8619402 0.84 HTT (0.33) HTTALDH1A1HPGDKDM4EMEN1
SCHEMBL8615494 0.84 SMN1; SMN2 (0.42) ALDH1A1HPGDKDM4EMEN1KMT2A
SCHEMBL8616047 0.84 ALDH1A1 (0.45) HTTALDH1A1HPGDKDM4EKMT2A
SCHEMBL8619083 0.84 CA2 (0.44) HTTALDH1A1HPGDKDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed