SCHEMBL8619638

SCHEMBL8619638

CCC(=O)c1cccc(N)c1C(=O)CC

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.44
HSD17B10 Q99714 5/20 0.44
MMP2 P08253 1/20 0.41
CFTR P13569 1/20 0.40
HSP90AB1 P08238 1/20 0.39
MEN1 O00255 1/20 0.38
CYP3A4 P08684 1/20 0.38
PTGS1 P23219 1/20 0.38
DRD3 P35462 1/20 0.38
KMT2A Q03164 1/20 0.38
KDM4E B2RXH2 6/20 0.38
POLB P06746 1/20 0.38
PDK2 Q15119 1/20 0.38
HPGD P15428 4/20 0.37
MAPT P10636 2/20 0.37
GAA P10253 1/20 0.37
CDC25B P30305 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
NSD2 O96028 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9559838 0.88 CYP3A4 (0.43) ALDH1A1HSD17B10MMP2CFTRHSP90AB1
SCHEMBL14632194 0.87 ALDH1A1 (0.41) ALDH1A1HSD17B10MMP2CFTRHSP90AB1
SCHEMBL9632452 0.82 ALDH1A1 (0.46) ALDH1A1HSD17B10MMP2CFTRHSP90AB1
SCHEMBL1207894 0.82 ALDH1A1 (0.58) ALDH1A1HSD17B10CFTRHSP90AB1MEN1
SCHEMBL29568750 0.82 ALDH1A1 (0.58) ALDH1A1HSD17B10CFTRHSP90AB1MEN1
SCHEMBL13181078 0.81 CES2 (0.48) ALDH1A1HSD17B10MEN1CYP3A4PTGS1
SCHEMBL11409639 0.81 ALDH1A1 (0.49) ALDH1A1HSD17B10MMP2CFTRHSP90AB1
Hydrochloric Acid SCHEMBL1567993 0.80 ALDH1A1 (0.56) ALDH1A1HSD17B10CFTRHSP90AB1MEN1
SCHEMBL10970621 0.79 HSP90AB1 (0.44) ALDH1A1HSD17B10MMP2HSP90AB1MEN1
SCHEMBL27635347 0.79 P2RX7 (0.43) ALDH1A1HSD17B10MMP2CFTRHSP90AB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5767121-A ANTIINFLAMMATORY AND -ARTHRITIC AGENTS; ANTIPYRETICS; ANALGESICS; ADHESION PROTEIN EXPRESSION AND CYCLOXYGENASE AND 5-LIPOXYGENASE INHIBITORS; IMMUNOSUPPRESSANTS AND -MODULATORS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-06-16 US disclosed
EP-0612729-B1 Pyridine derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1997-04-23 EP disclosed
US-5561147-A ANTIINFLAMMATORY AGENT, ANTIPYRETIC, ANALGESICS, ANTIALLERGENS, IMMUNOSUPPRESSANTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-10-01 US disclosed
US-5457106-A Antiinflammatory agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-10-10 US disclosed
US-5389658-A Administering as antipyretic, antiinflammatory, analgesic, antiallergic, or immunosupressive agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-02-14 US disclosed
EP-0612729-A2 Pyridine derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1994-08-31 EP disclosed
US-5246948-A Antiinflammatory, antipyretic, analgesic, antiallergic, immunosupressing or immunomodulating activity TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-09-21 US disclosed
EP-0522606-A2 Pyridine derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-01-13 EP disclosed