SCHEMBL8619903

SCHEMBL8619903

N=C(NC=O)Nc1cc(-c2ccccc2)nc2c(I)cccc12

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ACP1 P24666 3/20 0.39
ABCB1 P08183 1/20 0.38
ABCC1 P33527 1/20 0.38
ABCG2 Q9UNQ0 1/20 0.38
CYP2C9 P11712 1/20 0.38
ADORA3 P0DMS8 1/20 0.37
MEN1 O00255 1/20 0.37
GFER P55789 1/20 0.37
KMT2A Q03164 1/20 0.37
PDE4B Q07343 1/20 0.35
ADORA1 P30542 1/20 0.35
CHRNB2 P17787 1/20 0.35
CHRNB4 P30926 1/20 0.35
CHRNA3 P32297 1/20 0.35
CHRNA4 P43681 1/20 0.35
SLC2A1 P11166 1/20 0.35
PDE10A Q9Y233 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8615997 0.87 CCR6 (0.45) ACP1ABCB1ABCC1ABCG2CYP2C9
SCHEMBL8618767 0.86 MAPT (0.40) ACP1ABCB1ABCC1ABCG2CYP2C9
SCHEMBL8616699 0.86 ACP1 (0.39) ACP1ABCB1ABCC1ABCG2CYP2C9
SCHEMBL8613487 0.86 KDM4E (0.44) ACP1ABCB1ABCC1ABCG2CYP2C9
SCHEMBL8618998 0.84 ABCB1 (0.47) ACP1ABCB1ABCC1ABCG2ADORA3
SCHEMBL8617718 0.84 PDE10A (0.56) ACP1ABCB1ABCC1ABCG2GFER
SCHEMBL8617753 0.83 ACP1 (0.51) ACP1ABCB1ABCC1ABCG2MEN1
SCHEMBL8615310 0.83 MEN1 (0.41) ACP1ABCG2MEN1KMT2A
SCHEMBL8619728 0.83 KEAP1 (0.43) ACP1ABCB1ABCC1ABCG2
SCHEMBL8620687 0.81 PDE10A (0.45) ACP1MEN1KMT2AADORA1PDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed