SCHEMBL8619728

SCHEMBL8619728

CS(=O)(=O)Nc1cccc2c(NC(=N)NC=O)cc(-c3ccccc3)nc12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.43
GLO1 Q04760 3/20 0.40
CKS1B P61024 2/20 0.40
SKP2 Q13309 2/20 0.40
ALDH1A1 P00352 2/20 0.39
LMNA P02545 2/20 0.39
HSP90AA1 P07900 2/20 0.39
KDM4E B2RXH2 1/20 0.39
MAPT P10636 1/20 0.39
HPGD P15428 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
MMP2 P08253 2/20 0.39
ACP1 P24666 1/20 0.39
ABCB1 P08183 1/20 0.38
ABCC1 P33527 1/20 0.38
ABCG2 Q9UNQ0 1/20 0.38
ALOX15 P16050 1/20 0.38
HTT P42858 1/20 0.38
GAA P10253 1/20 0.36
THRB P10828 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8614752 0.90 ACP1 (0.36) MMP2ACP1ABCB1ABCC1ABCG2
SCHEMBL8617040 0.87 KEAP1 (0.41) KEAP1GLO1CKS1BSKP2MMP2
SCHEMBL8615114 0.87 ACP1 (0.36) MMP2ACP1ABCB1ABCC1ABCG2
SCHEMBL8618998 0.86 ABCB1 (0.47) ALDH1A1KDM4EMAPTHPGDNPSR1
SCHEMBL8620923 0.85 ALOX5AP (0.38)
SCHEMBL8613487 0.85 KDM4E (0.44) ALDH1A1LMNAKDM4EMAPTHPGD
SCHEMBL8615331 0.84 ALDH1A1 (0.41) KEAP1ALDH1A1LMNAHSP90AA1KDM4E
SCHEMBL8615997 0.84 CCR6 (0.45) ACP1ABCB1ABCC1ABCG2
SCHEMBL8618767 0.83 MAPT (0.40) ALDH1A1LMNAKDM4EMAPTHPGD
SCHEMBL8616699 0.83 ACP1 (0.39) KDM4EACP1ABCB1ABCC1ABCG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed