SCHEMBL8620067

SCHEMBL8620067

C=Cc1ccc(-c2ccccc2[N+](=O)[O-])cc1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.65
TDP1 Q9NUW8 2/20 0.65
ADAMTS4 O75173 1/20 0.42
PTPN1 P18031 1/20 0.41
S100A4 P26447 2/20 0.41
PTPRC P08575 1/20 0.41
TSHR P16473 2/20 0.41
SOS1 Q07889 1/20 0.41
HSD17B10 Q99714 2/20 0.40
GFER P55789 1/20 0.40
MGAM O43451 1/20 0.40
GAA P10253 1/20 0.40
SI P14410 1/20 0.40
MGAM2 Q2M2H8 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
TP53 P04637 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4373563 0.84 ALDH1A1 (0.67) ALDH1A1TDP1ADAMTS4PTPN1S100A4
SCHEMBL6747891 0.82 ALDH1A1 (0.74) ALDH1A1TDP1ADAMTS4PTPN1S100A4
SCHEMBL2958562 0.80 ALDH1A1 (0.92) ALDH1A1TDP1ADAMTS4PTPN1S100A4
Formaldehyde SCHEMBL28138834 0.80 ALDH1A1 (0.92) ALDH1A1TDP1ADAMTS4PTPN1S100A4
Benzene SCHEMBL28038982 0.79 ALDH1A1 (1.00) ALDH1A1TDP1ADAMTS4PTPN1S100A4
SCHEMBL30196067 0.79 ALDH1A1 (1.00) ALDH1A1TDP1ADAMTS4PTPN1S100A4
SCHEMBL44392 0.79 ALDH1A1 (1.00) ALDH1A1TDP1ADAMTS4PTPN1S100A4
SCHEMBL7821087 0.78 ALDH1A1 (0.74) ALDH1A1TDP1ADAMTS4PTPN1S100A4
SCHEMBL11792031 0.77 ALDH1A1 (0.88) ALDH1A1TDP1ADAMTS4PTPN1S100A4
Methane SCHEMBL2186810 0.77 ALDH1A1 (0.96) ALDH1A1TDP1ADAMTS4PTPN1S100A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0632017-B1 N-phenyl-2-cyano-3-hydroxy propenamides, their tautomeres and salts, their use as medicaments and compositions containing them HOECHST MARION ROUSSEL INC (FR) 1998-05-06 EP disclosed
US-5416112-A Antiinflammatory agents ROUSSEL UCLAF (FR) 1995-05-16 US disclosed
US-5385931-A Multistage formation of sulfonamides by reaction of esters and acyl halides, nitriding, reduction and sulfonylation to form cardiovascular compounds PIERRE FABRE MEDICAMENT (FR) 1995-01-31 US disclosed
EP-0632017-A1 N-phenyl-2-cyano-3-hydroxy propenamides, their tautomeres and salts, their use as medicaments and compositions containing them ROUSSEL UCLAF (FR) 1995-01-04 EP disclosed