SCHEMBL8620107

SCHEMBL8620107

Cc1ccccc1-c1cc(NC(=N)NC=O)c2ccc(O)cc2n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.37
ALDH1A1 P00352 7/20 0.37
HPGD P15428 5/20 0.37
KDM4E B2RXH2 5/20 0.37
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
MAPT P10636 3/20 0.36
ALOX12 P18054 1/20 0.36
MAPK10 P53779 1/20 0.36
ATM Q13315 1/20 0.36
POLB P06746 1/20 0.35
HSD17B10 Q99714 3/20 0.35
USP2 O75604 1/20 0.35
ERAP1 Q9NZ08 1/20 0.35
TACR3 P29371 2/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
GPR55 Q9Y2T6 1/20 0.34
GAA P10253 2/20 0.34
TP53 P04637 1/20 0.34
CYP1A2 P05177 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8614948 0.92 HTT (0.39) HTTALDH1A1HPGDKDM4EMEN1
SCHEMBL8620892 0.89 HTT (0.47) HTTALDH1A1HPGDKDM4EMEN1
SCHEMBL8615234 0.88 HTT (0.38) HTTALDH1A1HPGDKDM4EMEN1
SCHEMBL8613684 0.87 NPC1 (0.42) HTTALDH1A1HPGDKDM4EMEN1
SCHEMBL8619346 0.87 TACR3 (0.46) ALDH1A1HPGDKDM4EMAPTTACR3
SCHEMBL8615210 0.84 TACR3 (0.44) MEN1KMT2APOLBTACR3ACP1
SCHEMBL8619771 0.84 HTT (0.35) HTTALDH1A1HPGDKDM4EMEN1
SCHEMBL8613388 0.84 SMN1; SMN2 (0.39) HTTALDH1A1HPGDKDM4EMEN1
SCHEMBL8617771 0.84 ALDH1A1 (0.40) HTTALDH1A1HPGDKDM4EMAPT
SCHEMBL8617890 0.83 MEN1 (0.45) HTTALDH1A1HPGDMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed