SCHEMBL8624565

SCHEMBL8624565

CN(C)Cc1ccccc1C(=O)N1CCCN(CCC(c2ccccc2)c2ccccc2)CC1

nearest known ligand 0.48

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 16/20 0.48
CCR2 P41597 2/20 0.44
OPRM1 P35372 1/20 0.43
OPRL1 P41146 1/20 0.43
CHRM1 P11229 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6768750 0.83 HRH3 (0.55) CCR5CCR2CHRM1
SCHEMBL6770020 0.79 KMT2A (0.58) CCR2
SCHEMBL6768747 0.72 MEN1 (0.53) CCR2
SCHEMBL6765593 0.71 CCR2 (0.57) CCR5CCR2OPRM1OPRL1
SCHEMBL8572593 0.70 CCR2 (0.56) CCR5CCR2OPRM1OPRL1
SCHEMBL6703958 0.70 CCR5 (0.74) CCR5
SCHEMBL12333385 0.68 HRH4 (0.55) CHRM1
SCHEMBL8565906 0.68 CCR2 (0.54) CCR5CCR2OPRM1OPRL1
SCHEMBL8565792 0.68 CCR2 (0.54) CCR5CCR2OPRM1OPRL1
SCHEMBL15966084 0.68 KMT2A (0.68) CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997044329-A9 DIARYLALKYL CYCLIC DIAMINE DERIVATIVES AS CHEMOKINE RECEPTOR ANTAGONISTS 1998-03-12 WO disclosed